Synthesis of 1-indanones with a broad range of biological activity

Marika Turek, Dorota Szczęsna, Marek Koprowski and Piotr Bałczewski
Beilstein J. Org. Chem. 2017, 13, 451–494.

Cite the Following Article

Synthesis of 1-indanones with a broad range of biological activity
Marika Turek, Dorota Szczęsna, Marek Koprowski and Piotr Bałczewski
Beilstein J. Org. Chem. 2017, 13, 451–494.

How to Cite

Turek, M.; Szczęsna, D.; Koprowski, M.; Bałczewski, P. Beilstein J. Org. Chem. 2017, 13, 451–494. doi:10.3762/bjoc.13.48

Download Citation

Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window below.
Citation data in RIS format can be imported by all major citation management software, including EndNote, ProCite, RefWorks, and Zotero.

Presentation Graphic

Picture with graphical abstract, title and authors for social media postings and presentations.
Format: PNG Size: 779.6 KB Download

Citations to This Article

Up to 20 of the most recent references are displayed here.

Scholarly Works

  • Lan, S.; Zhang, W.; Gan, X. Novel 1-Indanone derivatives containing oxime and oxime ether moieties as immune activator to resist plant virus. Pest management science 2023, 79, 2686–2695. doi:10.1002/ps.7442
  • Inagaki, T.; Ando, T.; Sakurai, S.; Yamanaka, M.; Tobisu, M. Palladium-catalyzed addition of acylsilanes across alkynes via the activation of a C-Si bond. Chemical science 2023, 14, 2706–2712. doi:10.1039/d3sc00181d
  • Li, K.; Long, X.; Zhu, S. Photoredox/Nickel Dual Catalysis-Enabled Modular Synthesis of Arylallyl Alcohols with Acetylene as the Two-Carbon Synthon. ACS Catalysis 2023, 13, 2422–2431. doi:10.1021/acscatal.2c06178
  • Bansal, R.; Singh, R.; Rana, P. Synthesis, in silico Studies and Pharmacological Evaluation of a New Series of Indanone Derivatives as Anti-Parkinsonian and Anti-Alzheimer's Agents. Current computer-aided drug design 2023, 19, 94–107. doi:10.2174/1573409919666221129155110
  • Pigot, C.; Brunel, D.; Dumur, F. Indane-1,3-Dione: From Synthetic Strategies to Applications. Molecules (Basel, Switzerland) 2022, 27, 5976. doi:10.3390/molecules27185976
  • Sun, Y.; Li, Y.; Li, X.; Meng, L.; Zeng, Y. The role of halogen bonds in the catalytic mechanism of the iso-Nazarov cyclization reaction: a DFT study. Physical chemistry chemical physics : PCCP 2022, 24, 18877–18887. doi:10.1039/d2cp01913b
  • Negi, R.; Jena, T. K.; Jyoti; Tuti, N. K.; Anindya, R.; Khan, F. A. Solvent controlled synthesis of 2,3-diarylepoxy indenones and α-hydroxy diarylindanones and their evaluation as inhibitors of DNA alkylation repair. Organic & biomolecular chemistry 2022, 20, 5820–5835. doi:10.1039/d2ob00595f
  • Sambasiva Rao, Y. N.; Ghosh, P.; Mainkar, P. S.; Chandrasekhar, S. Access to Spiroindanolactones/lactams through an Aryne Insertion/Spirocyclization Strategy. Organic letters 2022, 24, 5372–5375. doi:10.1021/acs.orglett.2c02046
  • Ramesh, G.; Ramulu, B. V.; Balamurugan, R. Activation of o-Propargyl Alcohol Benzaldehydes under Acetalization Conditions for Intramolecular Electrophile Intercepted Meyer-Schuster Rearrangement. The Journal of organic chemistry 2022, 87, 8633–8647. doi:10.1021/acs.joc.2c00826
  • Bertero, N. M.; Apesteguía, C. R.; Marchi, A. J. Selective synthesis of 1-indanol by 1-indanone liquid-phase hydrogenation over metal-based catalysts: A LHHW kinetic approach. Chemical Engineering Science 2022, 254, 117629. doi:10.1016/j.ces.2022.117629
  • Sebastian, S.; Sylvestre, S.; Sundaraganesan, N.; Karthikeyan, B.; Silvan, S. Conformational analysis, molecular structure, spectroscopic, NBO, reactivity descriptors, wavefunction and molecular docking investigations of 5,6-dimethoxy-1-indanone: A potential anti Alzheimer's agent. Heliyon 2022, 8, e08821. doi:10.1016/j.heliyon.2022.e08821
  • Boukherrouba, E.; Larosa, C.; Nguyen, K.-A.; Caburet, J.; Lunven, L.; Bonnet, H.; Fortuné, A.; Boumendjel, A.; Boucherle, B.; Chierici, S.; Peuchmaur, M. Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers. European journal of medicinal chemistry 2022, 231, 114139. doi:10.1016/j.ejmech.2022.114139
  • Dorjay Lama, P.; Bhaskara Rao, L.; Sreenivasulu, C.; Ravi Kishore, D.; Satyanarayana, G. Single‐Column‐Based Heck Coupling, Condensation and Alkylation Strategy: Synthesis of 2‐Benzoyl‐2‐alkyl‐2,3‐dihydro‐1H‐inden‐1‐ones. ChemistrySelect 2021, 6, 13041–13045. doi:10.1002/slct.202102811
  • Cluzeau, J.; Nettekoven, U.; Kovacevic, M.; Časar, Z. Concise Six-Step Asymmetric Approach to Ramelteon from an Acetophenone Derivative Using Ir, Rh, Cu, and Ni Catalysis. The Journal of organic chemistry 2021, 87, 2129–2135. doi:10.1021/acs.joc.1c01614
  • Yang, B.; Li, S.-J.; Wang, Y.; Lan, Y.; Zhu, S. Hydrogen radical-shuttle (HRS)-enabled photoredox synthesis of indanones via decarboxylative annulation. Nature communications 2021, 12, 5257. doi:10.1038/s41467-021-25594-4
  • Meng, X.; Chen, D.; Rui, L.; Jiang, P.; Huang, S. Synthesis of 2-(Cyanomethyl)benzoic Esters via Carbon-Carbon Bond Cleavage of Indanones. The Journal of organic chemistry 2021, 86, 10852–10860. doi:10.1021/acs.joc.1c01131
  • Yu, K.-Y.; Deng, Y.-H.; Ge, X.-M.; An, X.-T.; Shu, P.-F.; Cao, Y.-X.; Zhao, X.-H.; Fan, C.-A. Tandem (2 + 2) Annulation/Retro-4π Electrocyclization/Imino-Nazarov Cyclization Reaction of p-Quinone Methides with Ynamides: Expeditious Construction of Functionalized Aminoindenes. Organic letters 2021, 23, 5885–5890. doi:10.1021/acs.orglett.1c02003
  • Park, S.; Lee, H.-K. Efficient kinetic resolution in the asymmetric transfer hydrogenation of 3-aryl-indanones: applications to a short synthesis of (+)-indatraline and a formal synthesis of (R)-tolterodine. RSC advances 2021, 11, 23161–23183. doi:10.1039/d1ra04538e
  • Yang, Y.; Wang, X.; Ye, X.; Wang, B.; Bao, X.; Wang, H. Advances of α-activated cyclic isothiocyanate for the enantioselective construction of spirocycles. Organic & biomolecular chemistry 2021, 19, 4610–4621. doi:10.1039/d1ob00564b
  • Olyaei, A.; Ebrahimi, S.; Sadeghpour, M. Convenient one-pot synthesis of some novel heteroaryl aminoindandione derivatives. Research on Chemical Intermediates 2021, 47, 2719–2730. doi:10.1007/s11164-021-04440-8
Other Beilstein-Institut Open Science Activities