Computational prediction of C–H hydricities and their use in predicting the regioselectivity of electron-rich C–H functionalisation reactions

  • Rasmus M. Borup,
  • Nicolai Ree and
  • Jan H. Jensen

Beilstein J. Org. Chem. 2026, 22, 603–610, doi:10.3762/bjoc.22.46

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Published 17 Apr 2026

Regioselective approach to 5-arylsulfonylisoxazoles and their antimicrobial activity

  • Artem S. Sazonov,
  • Dmitry A. Vasilenko,
  • Denis V. Porfiriev,
  • Yuri K. Grishin,
  • Rimma A. Gazzaeva,
  • Alisa P. Chernyshova,
  • Maxim A. Kryakvin,
  • Anna A. Baranova,
  • Vera A. Alferova and
  • Elena B. Averina

Beilstein J. Org. Chem. 2026, 22, 592–602, doi:10.3762/bjoc.22.45

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Published 17 Apr 2026

Design and synthesis of an erdafitinib-based selective FGFR2 degrader

  • Yumeng Jin,
  • Shidong Wang,
  • Sihan Pan,
  • Shuqi Huang,
  • Weichen Zhou,
  • Xiaohao Huang,
  • Lei Zheng and
  • Lingfeng Chen

Beilstein J. Org. Chem. 2026, 22, 583–591, doi:10.3762/bjoc.22.44

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Published 15 Apr 2026

Continuous-flow carbonyl hydrogenation under subatmospheric to atmospheric hydrogen pressure enabled by robust heterogeneous Pt–Fe catalysts

  • Hiroyuki Miyamura,
  • Ryosuke Kajiyama,
  • Shun-ya Onozawa,
  • Yoshihiro Kon and
  • Shū Kobayashi

Beilstein J. Org. Chem. 2026, 22, 575–582, doi:10.3762/bjoc.22.43

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Published 10 Apr 2026

Kinetic resolution of racemic planar-chiral vinylcymantrenes by molybdenum-catalyzed asymmetric metathesis dimerization

  • Haruna Imazu,
  • Hitoshi Izu,
  • Yasuhiro Ohki and
  • Masamichi Ogasawara

Beilstein J. Org. Chem. 2026, 22, 568–574, doi:10.3762/bjoc.22.42

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Published 31 Mar 2026

Molecular tweezer–peptide conjugates disrupt the protein–protein interaction between survivin and histone H3 essential in mitosis

  • Catherine Gsell,
  • Philipp Rebmann,
  • Karina Opara,
  • Christine Beuck,
  • Peter Bayer,
  • David Bier,
  • Ingrid R. Vetter and
  • Thomas Schrader

Beilstein J. Org. Chem. 2026, 22, 557–567, doi:10.3762/bjoc.22.41

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Published 27 Mar 2026

Experimental and DFT studies on the regioselective methanolysis of 5-azido-9-oxabicyclo[6.1.0]nonan-4-yl 4-nitrobenzoate isomers

  • İlknur Polat,
  • Selçuk Eşsiz and
  • Emine Salamci

Beilstein J. Org. Chem. 2026, 22, 547–556, doi:10.3762/bjoc.22.40

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Published 26 Mar 2026

Melifoliox B, a novel phloroglucin derivative isolated from Melicope barbigera (Rutaceae) and synthesis of new oxidation products from melifoliones A and B

  • Horst Weber,
  • Kim-Thao Tran-Cong,
  • Bernhard Mayer,
  • Guido J. Reiss,
  • Iryna S. Konovalova,
  • Marc S. Appelhans,
  • Kenneth R. Wood and
  • Claus M. Passreiter

Beilstein J. Org. Chem. 2026, 22, 535–546, doi:10.3762/bjoc.22.39

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Published 24 Mar 2026

Get a better glimpse on sequential photoreactions of trisnorbornadienes with 19F NMR spectroscopy

  • Julian Felix Maria Hebborn,
  • Ben Eric Merten,
  • Thomas Paululat and
  • Heiko Ihmels

Beilstein J. Org. Chem. 2026, 22, 527–534, doi:10.3762/bjoc.22.38

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Published 23 Mar 2026

Modern synthetic pathways towards eribulin and its subunits

  • Sebastian Dominik Graf

Beilstein J. Org. Chem. 2026, 22, 495–526, doi:10.3762/bjoc.22.37

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Published 19 Mar 2026
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