Supporting Information
| Supporting Information File 1: NMR and HRMS spectra of compounds 3, 4 and analytical HPLC spectra of purified (λ at 254 nm and 225 nm) as well as crude (λ at 225 nm), electrospray ionization mass spectra and high-resolution mass spectra for bioconjugates 13 and 17. | ||
| Format: PDF | Size: 714.9 KB | Download |
Cite the Following Article
Novel solid-phase strategy for the synthesis of ligand-targeted fluorescent-labelled chelating peptide conjugates as a theranostic tool for cancer
Sagnik Sengupta, Mena Asha Krishnan, Premansh Dudhe, Ramesh B. Reddy, Bishnubasu Giri, Sudeshna Chattopadhyay and Venkatesh Chelvam
Beilstein J. Org. Chem. 2018, 14, 2665–2679.
https://doi.org/10.3762/bjoc.14.244
How to Cite
Sengupta, S.; Krishnan, M. A.; Dudhe, P.; Reddy, R. B.; Giri, B.; Chattopadhyay, S.; Chelvam, V. Beilstein J. Org. Chem. 2018, 14, 2665–2679. doi:10.3762/bjoc.14.244
Download Citation
Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window
below.
Citation data in RIS format can be imported by all major citation management software, including EndNote,
ProCite, RefWorks, and Zotero.
Presentation Graphic
| Picture with graphical abstract, title and authors for social media postings and presentations. | ||
| Format: PNG | Size: 1.1 MB | Download |
Citations to This Article
Up to 20 of the most recent references are displayed here.
Scholarly Works
- Zyk, N. Y.; Garanina, A. S.; Plotnikova, E. A.; Ber, A. P.; Nimenko, E. A.; Dashkova, N. S.; Uspenskaia, A. A.; Shafikov, R. R.; Skvortsov, D. A.; Petrov, S. A.; Pankratov, A. A.; Zyk, N. V.; Majouga, A. G.; Beloglazkina, E. K.; Machulkin, A. E. Synthesis of Prostate-Specific Membrane Antigen-Targeted Bimodal Conjugates of Cytotoxic Agents and Antiandrogens and Their Comparative Assessment with Monoconjugates. International journal of molecular sciences 2023, 24, 11327. doi:10.3390/ijms241411327
- Zyk, N. Y.; Petrov, S. A.; Zavertkina, M. V.; Uspenskaya, A. A.; Krasnikov, P. A.; Dashkova, N. S.; Beloglazkina, E. K.; Majouga, A. G.; Zyk, N. V.; Machulkin, A. E. Choice of the optimal synthetic approach for the polypeptide ligands of prostatic specific membrane antigen preparation. Mendeleev Communications 2023, 33, 472–475. doi:10.1016/j.mencom.2023.06.010
- Petrov, S. A.; Zyk, N. Y.; Machulkin, A. E.; Beloglazkina, E. K.; Majouga, A. G. PSMA-targeted low-molecular double conjugates for diagnostics and therapy. European journal of medicinal chemistry 2021, 225, 113752. doi:10.1016/j.ejmech.2021.113752
- Krishnan, M. A.; Yadav, K.; Chelvam, V. Agarose Micro-Well Platform for Rapid Generation of Homogenous 3D Tumor Spheroids. Current protocols 2021, 1, e199. doi:10.1002/cpz1.199
- Krishnan, M. A.; Chelvam, V. Developing μSpherePlatform Using a Commercial Hairbrush: An Agarose 3D Culture Platform for Deep-Tissue Imaging of Prostate Cancer. ACS applied bio materials 2021, 4, 4254–4270. doi:10.1021/acsabm.1c00086
- Krishnan, M. A.; Yadav, K.; Roach, P. D.; Chelvam, V. A targeted near-infrared nanoprobe for deep-tissue penetration and imaging of prostate cancer. Biomaterials science 2021, 9, 2295–2312. doi:10.1039/d0bm01970d
- Balogh, B.; Ivánczi, M.; Nizami, B.; Beke-Somfai, T.; Mándity, I. M. ConjuPepDB: a database of peptide-drug conjugates. Nucleic acids research 2020, 49, D1102–D1112. doi:10.1093/nar/gkaa950
- Temperini, A.; Aiello, D.; Mazzotti, F.; Athanassopoulos, C. M.; De Luca, P.; Siciliano, C. 2,3-Diaminopropanols Obtained from d-Serine as Intermediates in the Synthesis of Protected 2,3-l-Diaminopropanoic Acid (l-Dap) Methyl Esters. Molecules (Basel, Switzerland) 2020, 25, 1313–1333. doi:10.3390/molecules25061313
- Sengupta, S.; Krishnan, M. A.; Pandit, A.; Dudhe, P.; Sharma, R.; Chelvam, V. Tyrosine-based asymmetric urea ligand for prostate carcinoma: Tuning biological efficacy through in silico studies. Bioorganic chemistry 2019, 91, 103154. doi:10.1016/j.bioorg.2019.103154
Patents
- CHELVAM VENKATESH; SENGUPTA SAGNIK; KRISHNAN MENA ASHA; PANDIT AMIT. SMALL MOLECULE INHIBITORS FOR EARLY DIAGNOSIS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN CANCERS AND NEURODEGENERATIVE DISEASES. US 20200164075 A1, May 28, 2020.
