Synthesis and herbicidal activities of aryloxyacetic acid derivatives as HPPD inhibitors

Scholarly Works

• Ferraroni, M. Nonheme mono- and dioxygenases. Metalloenzymes; Elsevier, 2024; pp 467–484. doi:10.1016/b978-0-12-823974-2.00028-0
• Cai, H.; Gan, X.; Jin, Z.; Hao, G. Carboxylic Acid Derivatives in Herbicide Development. Journal of agricultural and food chemistry 2023, 71, 9973–9993. doi:10.1021/acs.jafc.3c00951
• Niemczak, M.; Stachowiak, W.; Kaczmarek, D. K.; Grzanka, M.; Sobiech, Ł. A comprehensive study demonstrating the influence of the solvent composition on the phytotoxicity of compounds, as exemplified by 2,4-D-based ILs with a choline-type cation. Pest management science 2023, 79, 3602–3610. doi:10.1002/ps.7543
• Lin, H.-Y.; Dong, J.; Dong, J.; Yang, W.-C.; Yang, G.-F. Insights into 4-hydroxyphenylpyruvate dioxygenase-inhibitor interactions from comparative structural biology. Trends in biochemical sciences 2023, 48, 568–584. doi:10.1016/j.tibs.2023.02.006
• Sharma, S.; Singh, D.; Kumar, S.; Vaishali; Jamra, R.; Banyal, N.; Deepika; Malakar, C. C.; Singh, V. An efficient metal-free and catalyst-free C-S/C-O bond-formation strategy: synthesis of pyrazole-conjugated thioamides and amides. Beilstein journal of organic chemistry 2023, 19, 231–244. doi:10.3762/bjoc.19.22
• Dong, J.; Dong, J.; Yu, X.-H.; Yan, Y.-C.; Nan, J.-X.; Ye, B.-Q.; Yang, W.-C.; Lin, H.-Y.; Yang, G.-F. Discovery of Subnanomolar Inhibitors of 4-Hydroxyphenylpyruvate Dioxygenase via Structure-Based Rational Design. Journal of agricultural and food chemistry 2023, 71, 1170–1177. doi:10.1021/acs.jafc.2c06727
• Wang, J.-Y.; Zhao, L.-X.; Shi, J.; Gao, S.; Ye, F.; Fu, Y. Discovery of novel HPPD inhibitors based on a combination strategy of pharmacophore, consensus docking and molecular dynamics. Journal of Molecular Liquids 2022, 362, 119683. doi:10.1016/j.molliq.2022.119683
• Chotpatiwetchkul, W.; Chotsaeng, N.; Laosinwattana, C.; Charoenying, P. Structure-Activity Relationship Study of Xanthoxyline and Related Small Methyl Ketone Herbicides. ACS omega 2022, 7, 29002–29012. doi:10.1021/acsomega.2c02704
• Martins, F. A.; Daré, J. K.; Freitas, M. P. Computer-Assisted Proposition of Promising Aryloxyacetic Acid Derivatives as HPPD Inhibitors. Journal of agricultural and food chemistry 2022, 70, 8986–8993. doi:10.1021/acs.jafc.2c02954
• Shi, J.; Zhao, L.-X.; Wang, J.-Y.; Ye, T.; Wang, M.; Gao, S.; Ye, F.; Fu, Y. The novel 4-hydroxyphenylpyruvate dioxygenase inhibitors in vivo and in silico approach: 3D-QSAR analysis, molecular docking, bioassay and molecular dynamics. Arabian Journal of Chemistry 2022, 15, 103919. doi:10.1016/j.arabjc.2022.103919
• Zeng, H.; Zhang, W.; Wang, Z.; Geng, W.; Feng, G.; Gan, X. Novel Pyrazole Amides as Potential 4-Hydroxyphenylpyruvate Dioxygenase Inhibitors. Journal of agricultural and food chemistry 2022, 70, 7400–7411. doi:10.1021/acs.jafc.2c02123
• Governa, P.; Bernardini, G.; Braconi, D.; Manetti, F.; Santucci, A.; Petricci, E. Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations. Journal of agricultural and food chemistry 2022, 70, 6963–6981. doi:10.1021/acs.jafc.2c02010
• Agrwal, A.; Verma, A.; Chantola, N.; Verma, S.; Kasana, V. Synthesis, molecular docking and extensive structure activity relationship of substituted DHP derivatives: a new class of herbicides. Journal of environmental science and health. Part. B, Pesticides, food contaminants, and agricultural wastes 2022, 57, 379–420. doi:10.1080/03601234.2022.2062188
• Barber, D. M. A Competitive Edge: Competitor Inspired Scaffold Hopping in Herbicide Lead Optimization. Journal of agricultural and food chemistry 2022, 70, 11075–11090. doi:10.1021/acs.jafc.1c07910
• Song, H.-M.; Zhao, L.-X.; Zhang, S.-Q.; Ye, T.; Fu, Y.; Ye, F. Design, Synthesis, Structure-Activity Relationship, Molecular Docking, and Herbicidal Evaluation of 2-Cinnamoyl-3-Hydroxycyclohex-2-en-1-one Derivatives as Novel 4-Hydroxyphenylpyruvate Dioxygenase Inhibitors. Journal of agricultural and food chemistry 2021, 69, 12621–12633. doi:10.1021/acs.jafc.1c04621
• Mykhailiuk, P. K. Fluorinated Pyrazoles: From Synthesis to Applications. Chemical reviews 2020, 121, 1670–1715. doi:10.1021/acs.chemrev.0c01015
• Huang, H.; Zhang, J.-Q.; Liu, J.-M.; Wang, M.-M.; Shu, L.; Yan, Y.-L.; Zhan, X.-H.; Wang, P.; Huan, X.-T.; Dayong, Z. Discovery of novel benzofuran scaffold as 4-hydroxyphenylpyruvate dioxygenase inhibitors. Pest management science 2020, 77, 1409–1421. doi:10.1002/ps.6159
• Huang, H.; Wang, M.-M.; Shu, L.; Yan, Y.-L.; Zhang, J.-Q.; Liu, J.-M.; Zhan, X.-H.; Dayong, Z. Discovery of novel arylthioacetic acid derivatives as 4-hydroxyphenylpyruvate dioxygenase inhibitors. Pest management science 2020, 76, 4112–4122. doi:10.1002/ps.5967

Explore citations to this article at