Free-radical cyclization approach to polyheterocycles containing pyrrole and pyridine rings

Ivan P. Mosiagin,
Olesya A. Tomashenko,
Dar’ya V. Spiridonova,
Mikhail S. Novikov,
Sergey P. Tunik and
Alexander F. Khlebnikov

Full Research Paper
Published 23 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1490–1498, doi:10.3762/bjoc.17.105

Full Text

Cascade intramolecular Prins/Friedel–Crafts cyclization for the synthesis of 4-aryltetralin-2-ols and 5-aryltetrahydro-5H-benzo[7]annulen-7-ols

Jie Zheng,
Shuyu Meng and
Quanrui Wang

Full Research Paper
Published 22 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1481–1489, doi:10.3762/bjoc.17.104

Full Text

Co-crystallization of an organic solid and a tetraaryladamantane at room temperature

Fabian Rami,
Jan Nowak,
Felix Krupp,
Wolfgang Frey and
Clemens Richert

Letter
Published 21 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1476–1480, doi:10.3762/bjoc.17.103

Full Text

Iodine-catalyzed electrophilic substitution of indoles: Synthesis of (un)symmetrical diindolylmethanes with a quaternary carbon center

Thanigaimalai Pillaiyar,
Masoud Sedaghati,
Andhika B. Mahardhika,
Lukas L. Wendt and
Christa E. Müller

Full Research Paper
Published 18 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1464–1475, doi:10.3762/bjoc.17.102

Full Text

Synthesis of 1-indolyl-3,5,8-substituted γ-carbolines: one-pot solvent-free protocol and biological evaluation

Premansh Dudhe,
Mena Asha Krishnan,
Kratika Yadav,
Diptendu Roy,
Krishnan Venkatasubbaiah,
Biswarup Pathak and
Venkatesh Chelvam

Letter
Published 17 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1453–1463, doi:10.3762/bjoc.17.101

Full Text

Organocatalytic asymmetric Michael/acyl transfer reaction between α-nitroketones and 4-arylidenepyrrolidine-2,3-diones

Chandrakanta Parida and
Subhas Chandra Pan

Full Research Paper
Published 14 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1447–1452, doi:10.3762/bjoc.17.100

Full Text

Total synthesis of ent-pavettamine

Memory Zimuwandeyi,
Manuel A. Fernandes,
Amanda L. Rousseau and
Moira L. Bode

Full Research Paper
Published 10 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1440–1446, doi:10.3762/bjoc.17.99

Full Text

Double-headed nucleosides: Synthesis and applications

Vineet Verma,
Jyotirmoy Maity,
Vipin K. Maikhuri,
Ritika Sharma,
Himal K. Ganguly and
Ashok K. Prasad

Review
Published 08 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1392–1439, doi:10.3762/bjoc.17.98

Full Text

Analogs of the carotane antibiotic fulvoferruginin from submerged cultures of a Thai Marasmius sp.

Birthe Sandargo,
Leon Kaysan,
Rémy B. Teponno,
Christian Richter,
Benjarong Thongbai,
Frank Surup and
Marc Stadler

Full Research Paper
Published 04 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1385–1391, doi:10.3762/bjoc.17.97

Full Text

Design, synthesis and photophysical properties of novel star-shaped truxene-based heterocycles utilizing ring-closing metathesis, Clauson–Kaas, Van Leusen and Ullmann-type reactions as key tools

Shakeel Alvi and
Rashid Ali

Full Research Paper
Published 02 Jun 2021

Beilstein J. Org. Chem. 2021, 17, 1374–1384, doi:10.3762/bjoc.17.96

Full Text

Supporting Information File 1: Detailed experimental protocols and supporting ¹H, ¹³C NMR, LC–MS characterization data and spectra for all compounds.
Format: PDF	Size: 8.6 MB	Download

Article Citation
Download RIS (Reference Manager)	Download BIB (BIBTEX)
Cited References
Download RIS (Reference Manager)	Download BIB (BIBTEX)

Novel library synthesis of 3,4-disubstituted pyridin-2(1H)-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature

Supporting Information

References

Presentation Graphic

Latest Articles

Free-radical cyclization approach to polyheterocycles containing pyrrole and pyridine rings

Cascade intramolecular Prins/Friedel–Crafts cyclization for the synthesis of 4-aryltetralin-2-ols and 5-aryltetrahydro-5H-benzo[7]annulen-7-ols

Co-crystallization of an organic solid and a tetraaryladamantane at room temperature

Iodine-catalyzed electrophilic substitution of indoles: Synthesis of (un)symmetrical diindolylmethanes with a quaternary carbon center

Synthesis of 1-indolyl-3,5,8-substituted γ-carbolines: one-pot solvent-free protocol and biological evaluation

Organocatalytic asymmetric Michael/acyl transfer reaction between α-nitroketones and 4-arylidenepyrrolidine-2,3-diones

Total synthesis of ent-pavettamine

Double-headed nucleosides: Synthesis and applications

Analogs of the carotane antibiotic fulvoferruginin from submerged cultures of a Thai Marasmius sp.

Design, synthesis and photophysical properties of novel star-shaped truxene-based heterocycles utilizing ring-closing metathesis, Clauson–Kaas, Van Leusen and Ullmann-type reactions as key tools

Latest Thematic Issues

GlycoBioinformatics

Molecular recognition

Organo-fluorine chemistry V

Celebrating the role of chemistry in the success of oligonucleotides as therapeutics

Chemical ecology

Advances in photoredox catalysis

Green chemistry II

C–H functionalization for materials science

Medicinal chemistry and drug discovery in an opening era

Other Beilstein-Institut Open Science Activities

Keep Informed