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Cite the Following Article
β-Lactamase inhibition profile of new amidine-substituted diazabicyclooctanes
Zafar Iqbal, Lijuan Zhai, Yuanyu Gao, Dong Tang, Xueqin Ma, Jinbo Ji, Jian Sun, Jingwen Ji, Yuanbai Liu, Rui Jiang, Yangxiu Mu, Lili He, Haikang Yang and Zhixiang Yang
Beilstein J. Org. Chem. 2021, 17, 711–718.
https://doi.org/10.3762/bjoc.17.60
How to Cite
Iqbal, Z.; Zhai, L.; Gao, Y.; Tang, D.; Ma, X.; Ji, J.; Sun, J.; Ji, J.; Liu, Y.; Jiang, R.; Mu, Y.; He, L.; Yang, H.; Yang, Z. Beilstein J. Org. Chem. 2021, 17, 711–718. doi:10.3762/bjoc.17.60
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Scholarly Works
- Fatima, N.; Khalid, S.; Rasool, N.; Imran, M.; Parveen, B.; Kanwal, A.; Irimie, M.; Ciurea, C. I. Approachable Synthetic Methodologies for Second-Generation β-Lactamase Inhibitors: A Review. Pharmaceuticals (Basel, Switzerland) 2024, 17, 1108. doi:10.3390/ph17091108
- Zainal Abidin, A.; Norrrahim, M. N. F.; Mohamed Shakrin, N. N. S.; Ibrahim, B.; Abdullah, N.; Abdul Rashid, J. I.; Mohd Kasim, N. A.; Ahmad Shah, N. A. Amidine containing compounds: Antimicrobial activity and its potential in combating antimicrobial resistance. Heliyon 2024, 10, e32010. doi:10.1016/j.heliyon.2024.e32010
- He, L.; Yang, H.; Sun, J.; Zhai, L.; Ji, J.; Ma, X.; Tang, D.; Mu, Y.; Wang, L.; Iqbal, Z.; Yang, Z. Synthesis and β-Lactamase Inhibition Activity of Diazabicyclooctane Derivatives in Combination with Imipenem. Russian Journal of General Chemistry 2022, 92, 2888–2898. doi:10.1134/s1070363222120428
- Sun, J.; He, L.; Ji, J.; Zhai, L.; Ji, J.; Ma, X.; Tang, D.; Mu, Y.; Gao, Y.; Wang, L.; Yang, H.; Iqbal, Z.; Yang, Z. Synergistic Antibacterial Activity of Meropenem and Imipenem in Combination with Diazabicyclooctane Derivatives. Russian Journal of General Chemistry 2022, 92, 2070–2081. doi:10.1134/s1070363222100218
- Lijuan Zhai; Sun, J.; Ji, J.; He, L.; Gao, Y.; Ji, J.; Liu, Y.; Mu, Y.; Ma, X.; Tang, D.; Yang, H.; Iqbal, Z.; Yang, Z. Synthesis and β-Lactamase Inhibition Activity of Imidates of Diazabicyclooctane. Russian Journal of Bioorganic Chemistry 2022, 48, 1059–1067. doi:10.1134/s1068162022050120
- Iqbal, Z.; Sun, J.; Yang, H.; Ji, J.; He, L.; Zhai, L.; Ji, J.; Zhou, P.; Tang, D.; Mu, Y.; Wang, L.; Yang, Z. Recent Developments to Cope the Antibacterial Resistance via β-Lactamase Inhibition. Molecules (Basel, Switzerland) 2022, 27, 3832. doi:10.3390/molecules27123832
- Liu, Y.; Ji, J.; Sun, J.; He, L.; Gao, Y.; Zhai, L.; Ji, J.; Ma, X.; Mu, Y.; Tang, D.; Yang, H.; Iqbal, Z.; Yang, Z. Substituted-amidine derivatives of diazabicyclooctane as prospective β-lactamase inhibitors. Monatshefte für Chemie - Chemical Monthly 2022, 153, 301–309. doi:10.1007/s00706-021-02888-3
- Ji, J.; Zhai, L.; Sun, J.; He, L.; Ji, J.; Ma, X.; Liu, Y.; Tang, D.; Mu, Y.; Gao, Y.; Yang, H.; Iqbal, Z.; Yang, Z. Sulfonylamidine-substituted derivatives of avibactam: Synthesis and antibacterial activity. Journal of Heterocyclic Chemistry 2021, 58, 2390–2394. doi:10.1002/jhet.4360
Patents
- YANG ZHIXIANG; YANG HAIKANG; JI JINBO; ZHAI LIJUAN; SUN JIAN; JI JINGWEN; HE LILI; TANG DONG; IQBAL ZAFAR; LIU YUANBAI; MU YANGXIU; MA XUEQIN; YU JIANQIANG. Sulfonylamidine substituted compounds and their use as beta-lactamase inhibitors. US 12410166 B2, Sept 9, 2025.
- YANG ZHIXIANG; YANG HAIKANG; JI JINBO; ZHAI LIJUAN; SUN JIAN; JI JINGWEN; HE LILI; TANG DONG; IQBAL ZAFAR; LIU YUANBAI; MU YANGXIU; MA XUEQIN; YU JIANQIANG. SULFONYLAMIDINE SUBSTITUTED COMPOUNDS AND THEIR USE AS BETA-LACTAMASE INHIBITORS. US 20240132488 A1, April 25, 2024.
- YANG ZHIXIANG; YANG HAIKANG; JI JINBO; ZHAI LIJUAN; SUN JIAN; JI JINGWEN; HE LILI; TANG DONG; IQBAL ZAFAR; LIU YUANBAI; MU YANGXIU; MA XUEQIN; YU JIANQIANG. SULFONYLAMIDINE SUBSTITUTED COMPOUNDS AND THEIR USE AS BETA-LACTAMASE INHIBITORS. WO 2022233181 A1, Nov 10, 2022.
