Synthetic accesses to biguanide compounds

Oleksandr Grytsai, Cyril Ronco and Rachid Benhida
Beilstein J. Org. Chem. 2021, 17, 1001–1040. https://doi.org/10.3762/bjoc.17.82

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Synthetic accesses to biguanide compounds
Oleksandr Grytsai, Cyril Ronco and Rachid Benhida
Beilstein J. Org. Chem. 2021, 17, 1001–1040. https://doi.org/10.3762/bjoc.17.82

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Grytsai, O.; Ronco, C.; Benhida, R. Beilstein J. Org. Chem. 2021, 17, 1001–1040. doi:10.3762/bjoc.17.82

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  • Shi, X.; Zhang, R.; Sand, W.; Mathivanan, K.; Zhang, Y.; Wang, N.; Duan, J.; Hou, B. Comprehensive Review on the Use of Biocides in Microbiologically Influenced Corrosion. Microorganisms 2023, 11, 2194. doi:10.3390/microorganisms11092194
  • Makotchenko, E. V.; Yu. Kharlamova, V.; Baidina, I. A.; Bardina, E. E.; Korolkov, I. V.; Mironov, I. V.; Gushchin, A. L. Synthesis, crystal structure and solution studies of gold(III) complexes with 1,1-dimethylbiguanide. Inorganica Chimica Acta 2023, 552, 121496. doi:10.1016/j.ica.2023.121496
  • Koneshlou, T.; Rouhani, M.; Saeidian, H.; Aliabad, J. M. Biguanide-dihydropyrimidine dual scaffolds with impressive basicities according to DFT calculations. Computational and Theoretical Chemistry 2023, 1225, 114178. doi:10.1016/j.comptc.2023.114178
  • Bi, C.; Wang, Y.; He, C.; Baran, P. S. Enantioselective Total Synthesis of (+)-KB343. Journal of the American Chemical Society 2023, 145, 7753–7757. doi:10.1021/jacs.3c01991
  • Gungor, O.; Kose, M. Design, synthesis, biological evaluation and molecular docking of cyclic biguanidine compounds as cholinesterase inhibitors. Journal of biomolecular structure & dynamics 2022, 41, 10885–10899. doi:10.1080/07391102.2022.2158945
  • Farwa, U.; Raza, M. A. Heterocyclic compounds as a magic bullet for diabetes mellitus: a review. RSC advances 2022, 12, 22951–22973. doi:10.1039/d2ra02697j
  • Rios-Valenciana, E. E.; Menezes, O.; Niu, X.-Z.; Romero, J.; Root, R. A.; Chorover, J.; Sierra-Alvarez, R.; Field, J. A. Reductive transformation of the insensitive munitions compound nitroguanidine by different iron-based reactive minerals. Environmental pollution (Barking, Essex : 1987) 2022, 309, 119788. doi:10.1016/j.envpol.2022.119788
  • Güngör, Ö.; Köse, M. Design, synthesis and biological evaluation of biguanids and biguanid-sulfonamides as cholinesterase inhibitors. Journal of Molecular Structure 2022, 1260, 132817. doi:10.1016/j.molstruc.2022.132817
  • Grytsai, O.; Myrgorodska, I.; Rocchi, S.; Ronco, C.; Benhida, R. Biguanides drugs: Past success stories and promising future for drug discovery. European journal of medicinal chemistry 2021, 224, 113726. doi:10.1016/j.ejmech.2021.113726
  • Grytsai, O.; Gonçalves, L. C. P.; Bardovskyi, R.; Hamouda-Tekaya, N.; Rocchi, S.; Ronco, C.; Benhida, R. Arylbiamidines: synthesis and structural studies en route to anticancer applications. New Journal of Chemistry 2021, 45, 11893–11897. doi:10.1039/d1nj01943k

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