Efficient and improved synthesis of Telmisartan

A. Sanjeev Kumar, Samir Ghosh and G. N. Mehta
Beilstein J. Org. Chem. 2010, 6, No. 25. https://doi.org/10.3762/bjoc.6.25

Cite the Following Article

Efficient and improved synthesis of Telmisartan
A. Sanjeev Kumar, Samir Ghosh and G. N. Mehta
Beilstein J. Org. Chem. 2010, 6, No. 25. https://doi.org/10.3762/bjoc.6.25

How to Cite

Kumar, A. S.; Ghosh, S.; Mehta, G. N. Beilstein J. Org. Chem. 2010, 6, No. 25. doi:10.3762/bjoc.6.25

Download Citation

Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window below.
Citation data in RIS format can be imported by all major citation management software, including EndNote, ProCite, RefWorks, and Zotero.

Citations to This Article

Up to 20 of the most recent references are displayed here.

Scholarly Works

  • Dhibar, M.; Chakraborty, S.; Basak, S.; Pattanayak, P.; Chatterjee, T.; Ghosh, B.; Raafat, M.; Abourehab, M. A. S. Critical Analysis and Optimization of Stoichiometric Ratio of Drug-Coformer on Cocrystal Design: Molecular Docking, In Vitro and In Vivo Assessment. Pharmaceuticals (Basel, Switzerland) 2023, 16, 284. doi:10.3390/ph16020284
  • Patil, S.; M, P. K.; Chadar, R.; Ramar, S.; Prasad, A.; Koppula, P.; Koppula, S. Evaluation, Method Development, and Validation for Content Determination of Potential Genotoxic Impurities (PGIs) at the TTC Level in Telmisartan API. Organic Process Research & Development 2021, 25, 1391–1401. doi:10.1021/acs.oprd.1c00086
  • Ferlin, F.; Lanari, D.; Vaccaro, L. Sustainable flow approaches to active pharmaceutical ingredients. Green Chemistry 2020, 22, 5937–5955. doi:10.1039/d0gc02404j
  • Zhang, J.; Li, R.; Fuqiang, Z.; Changliang, S.; Shen, J. An improved synthesis of telmisartan via the copper-catalyzed cyclization of o -haloarylamidines. RSC advances 2020, 10, 13717–13721. doi:10.1039/d0ra00886a
  • Martínez, V. R.; Aguirre, M. V.; Todaro, J. S.; Ferrer, E. G.; Williams, P. A. Improvement of the Anticancer Activities of Telmisartan by Zn(II) Complexation and Mechanisms of Action. Biological trace element research 2019, 197, 454–463. doi:10.1007/s12011-019-02013-w
  • Gund, S. H.; Balsane, K. E.; Nagarkar, J. M. Desulfinylative Pd-catalyzed coupling reaction of arenediazonium salt with aryl sulfinates to give unsymmetrical biaryls. Tetrahedron Letters 2017, 58, 2936–2939. doi:10.1016/j.tetlet.2017.06.045
  • Rodríguez-Lara, S. Q.; Cardona-Muñoz, E. G.; Ramírez-Lizardo, E. J.; Totsuka-Sutto, S. E.; Castillo-Romero, A.; Garcia-Cobian, T. A.; García-Benavides, L. Alternative Interventions to Prevent Oxidative Damage following Ischemia/Reperfusion. Oxidative medicine and cellular longevity 2016, 2016, 7190943. doi:10.1155/2016/7190943
  • Cao, Y.; Shi, L.-L.; Cao, Q.-R.; Yang, M.; Cui, J.-H. In-Vitro Characterization and Oral Bioavailability of Organic Solvent-free Solid Dispersions Containing Telmisartan. Iranian journal of pharmaceutical research : IJPR 2016, 15, 385–394.
  • Porta, R.; Benaglia, M.; Puglisi, A. Flow Chemistry: Recent Developments in the Synthesis of Pharmaceutical Products. Organic Process Research & Development 2015, 20, 2–25. doi:10.1021/acs.oprd.5b00325
  • Martin, A. D.; Siamaki, A. R.; Belecki, K.; Gupton, B. F. A convergent approach to the total synthesis of telmisartan via a Suzuki cross-coupling reaction between two functionalized benzimidazoles. The Journal of organic chemistry 2015, 80, 1915–1919. doi:10.1021/jo5025333
  • Santra, S.; Hota, P. K.; Bhattacharyya, R.; Bera, P.; Ghosh, P.; Mandal, S. K. Palladium Nanoparticles on Graphite Oxide: A Recyclable Catalyst for the Synthesis of Biaryl Cores. ACS Catalysis 2013, 3, 2776–2789. doi:10.1021/cs400468h
  • Meti, G. Y.; Kamble, R. R.; Biradar, D. B.; Margankop, S. B. Synthesis of biphenyl derivatives as ACE and α-amylase inhibitors. Medicinal Chemistry Research 2013, 22, 5868–5877. doi:10.1007/s00044-013-0574-8
  • Yan, P.-C.; Guoliang, Z.; Xie, J.-H.; Xiangdong, Z.; Zhou, Q.-L.; Yuanqiang, L.; Shen, W.-H.; Daqing, C. Industrial Scale-Up of Enantioselective Hydrogenation for the Asymmetric Synthesis of Rivastigmine. Organic Process Research & Development 2013, 17, 307–312. doi:10.1021/op3003147
Other Beilstein-Institut Open Science Activities