Synthesis of the calcilytic ligand NPS 2143

Henrik Johansson, Thomas Cailly, Alex Rojas Bie Thomsen, Hans Bräuner-Osborne and Daniel Sejer Pedersen

Beilstein J. Org. Chem. 2013, 9, 1383–1387. https://doi.org/10.3762/bjoc.9.154

Supporting Information

1H and 13C NMR spectra and HPLC chromatograms for compounds 3, 4, 5, 6, 8, and 16. Chromatograms from chiral HPLC analysis of rac-3 and (R)-3 and experimental details for the pharmacological characterisation for (R)-3.

Supporting Information File 1: Experimental procedures and full characterisation of the calcilytic ligand NPS 2143.
Format: PDF Size: 1.6 MB Download

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