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1 article(s) from Farkas, Viktor

Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin–GnRH-III conjugates developed for targeted drug delivery

Sabine Schuster,
Beáta Biri-Kovács,
Bálint Szeder,
Viktor Farkas,
László Buday,
Zsuzsanna Szabó,
Gábor Halmos and
Gábor Mező

Beilstein J. Org. Chem. 2018, 14, 756–771, doi:10.3762/bjoc.14.64

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Scheme 1: Syntheses of GnRH-III–[(⁴Lys(Bu)/⁴Ser, ⁶Aaa, ⁸Lys(Dau=Aoa)] bioconjugates. a) (1) 2% hydrazine in D...

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Figure 1: Far-UV ECD spectra of GnRH-III and its drug conjugates in water (GnRH-III solid, K1 dash, K2 dot, 1...

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Figure 2: Degradation of the GnRH-III bioconjugates by rat liver lysosomal homogenate. A) Cleavage sites prod...

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Figure 3: Cytostatic effect of the GnRH-III bioconjugates at different concentrations on A) HT-29 and B) MCF-...

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Figure 4: Cellular uptake of the GnRH-III bioconjugates at different concentrations on A) HT-29 and B) MCF-7 ...

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Figure 5: Cellular uptake of bioconjugate K2 (40 µM) visualized by confocal laser scanning microscopy (CLSM) ...

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Figure 6: Competitive inhibition of the GnRH-R on MCF-7 cells. Cellular uptake of the GnRH-III bioconjugate K2...

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Published 04 Apr 2018

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