N-Propargylamines: versatile building blocks in the construction of thiazole cores

Scholarly Works

• Samiee Paghaleh, E.; Kolvari, E.; Seidi, F.; Dashtian, K. Eco-friendly and sustainable basil seed hydrogel-loaded copper hydroxide-based catalyst for the synthesis of propargylamines and tetrazoles. Nanoscale advances 2024, 6, 960–972. doi:10.1039/d3na01085f
• Sadashiva, M. P.; Singh, K. R.; Santhosh, C.; Sheela, K. Regioselective Synthesis of 2,4- and 2,5-Disubstituted 1,3-Thiazoles from 2-Oxo-2-(amino)ethanedithioates via Base-Catalyzed Cyclization. Synthesis 2023, 56, 878–886. doi:10.1055/a-2210-6357
• Ramirez, N. P.; Waser, J. Copper (I)‐BOX Catalyzed Asymmetric 3‐Component Reaction for the Synthesis of Trifluoromethylated Propargylic Ethers and Anilines**. Angewandte Chemie 2023, 135. doi:10.1002/ange.202305776
• Ramirez, N. P.; Waser, J. Copper (I)-BOX Catalyzed Asymmetric 3-Component Reaction for the Synthesis of Trifluoromethylated Propargylic Ethers and Anilines. Angewandte Chemie (International ed. in English) 2023, 62, e202305776. doi:10.1002/anie.202305776
• Li, C.; Liao, M.; He, Z.; Chen, Y.; Mai, J.; Dong, R.; Chen, J.; Chen, L. Metal‐Free Oxidative Cross‐Dehydrogenative Coupling of Alkenes with Thiophenols. ChemistrySelect 2023, 8. doi:10.1002/slct.202300845
• Pharande, P. S.; Rashinkar, G. S.; Pore, D. M. Silica-grafted DBU-supported NiCl2: a sustainable heterogeneous catalyst for A3 coupling. Research on Chemical Intermediates 2023, 49, 2359–2382. doi:10.1007/s11164-023-04980-1
• Narra, R. R.; Unnithan, V. G.; Wong, T. H.; Guo, Z. Thiamine carbene liganded gold(i) chloride catalyzes an efficient aldehyde–alkyne–amine coupling reaction in water. Green Chemistry 2023, 25, 1920–1924. doi:10.1039/d2gc04851e
• Bhoraniya, R. B.; Modha, S. G. Propargyl Amines: Versatile Building Blocks in Post-Ugi Transformations. ChemistryOpen 2023, 12, e202200223. doi:10.1002/open.202200223
• Singh, A.; Malhotra, D.; Singh, K.; Chadha, R.; Bedi, P. M. S. Thiazole derivatives in medicinal chemistry: Recent advancements in synthetic strategies, structure activity relationship and pharmacological outcomes. Journal of Molecular Structure 2022, 1266, 133479. doi:10.1016/j.molstruc.2022.133479
• Kaur, N.; Sharma, K.; Grewal, P. Synthesis of heterocycles from urea and its derivatives. Synthetic Communications 2022, 52, 1867–1899. doi:10.1080/00397911.2022.2117630
• Shehzadi, S. A.; Saeed, A.; Perveen, F.; Channar, P. A.; Arshad, I.; Abbas, Q.; Kalsoom, S.; Yousaf, S.; Simpson, J. Identification of two novel thiazolidin-2-imines as tyrosinase inhibitors: synthesis, crystal structure, molecular docking and DFT studies. Heliyon 2022, 8, e10098. doi:10.1016/j.heliyon.2022.e10098
• Wang, Z.; Yang, B. General Strategies for Rational Design and Discovery of Multitarget Drugs. Polypharmacology; Springer International Publishing, 2022; pp 677–736. doi:10.1007/978-3-031-04998-9_18
• Cirujano, F. G.; Dhakshinamoorthy, A. Supported metals on porous solids as heterogeneous catalysts for the synthesis of propargylamines. New Journal of Chemistry 2022, 46, 1469–1482. doi:10.1039/d1nj05091e
• Shehzadi, S. A.; Saeed, A.; Perveen, F.; Channar, P. A.; Arshad, M. I.; Abbas, Q.; Kalsoom, S.; Yousaf, S.; Simpson, J. Identification of Two Novel Thiazolidin-2-Imines as Tyrosinase Inhibitors: Synthesis, Crystal Structure, Molecular Docking and DFT Studies. SSRN Electronic Journal 2022. doi:10.2139/ssrn.4129847
• Cao, Y.; Ahmadi, R.; Poor Heravi, M. R.; Issakhov, A.; Ebadi, A. G.; Vessally, E. Recent trends in dehydroxylative trifluoro-methylation, -methoxylation, -methylthiolation, and -methylselenylation of alcohols. RSC advances 2021, 11, 39593–39606. doi:10.1039/d1ra05018d
• Al-Mubaddel, F. S.; Karimi, M.; Sadeghi, S.; Gavinehroudi, R. G.; Mohebali, H.; Mahjoub, A. R.; Marzouki, R.; Ouni, M. H. E.; Heydari, A. Amino acid-assisted ferrite/MOF composite formation for visible-light induced photocatalytic cascade C=C aerobic oxidative cleavage functionalization. Molecular Catalysis 2021, 516, 111949. doi:10.1016/j.mcat.2021.111949
• Zhang, C.-C.; Chen, L.-J.; Shen, B.-C.; Xie, H.-D.; Li, W.; Sun, Z.-W. Enantioselective decarboxylative Mannich reaction of β-keto acids with C-alkynyl N-Boc N,O-acetals: access to chiral β-keto propargylamines. Organic & biomolecular chemistry 2021, 19, 8607–8612. doi:10.1039/d1ob01555a
• Klintworth, R.; Morgans, G. L.; Scalzullo, S. M.; de Koning, C. B.; van Otterlo, W. A. L.; Michael, J. P. Silica gel and microwave-promoted synthesis of dihydropyrrolizines and tetrahydroindolizines from enaminones. Beilstein journal of organic chemistry 2021, 17, 2543–2552. doi:10.3762/bjoc.17.170
• Cao, Y.; Abdolmohammadi, S.; Ahmadi, R.; Issakhov, A.; Ebadi, A. G.; Vessally, E. Direct synthesis of sulfenamides, sulfinamides, and sulfonamides from thiols and amines. RSC advances 2021, 11, 32394–32407. doi:10.1039/d1ra04368d
• Lim, J.; Lee, S. Metal-Free Doubly Decarboxylative Three-Component Reaction: Synthesis of Propargyl Amines. Asian Journal of Organic Chemistry 2021, 10, 2530–2533. doi:10.1002/ajoc.202100454

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