Synthesis of pyrazolopyrimidinones using a “one-pot” approach under microwave irradiation

Scholarly Works

• Gao, G.; Li, Z. Metal-free synthesis of ketonitrilesviaC–F bond cleavage. New Journal of Chemistry 2023, 47, 6171–6175. doi:10.1039/d2nj06338g
• Constantin, T.; Górski, B.; Tilby, M. J.; Chelli, S.; Juliá, F.; Llaveria, J.; Gillen, K. J.; Zipse, H.; Lakhdar, S.; Leonori, D. Halogen-atom and group transfer reactivity enabled by hydrogen tunneling. Science (New York, N.Y.) 2022, 377, 1323–1328. doi:10.1126/science.abq8663
• Pravin, N.; Jozwiak, K. Effects of Linkers and Substitutions on Multitarget Directed Ligands for Alzheimer's Diseases: Emerging Paradigms and Strategies. International journal of molecular sciences 2022, 23, 6085. doi:10.3390/ijms23116085
• Kodonidi, I. P.; Anenko, D. S.; Pozdnyakov, D. I. Synthesis and Action of N-acylphenylacetamides and N-acyl-β-ketoamides on the Central Nervous System. Drug development & registration 2022, 11, 40–49. doi:10.33380/2305-2066-2022-11-1-40-49
• Feng, Y.; He, J.; Wei, Y.; Tang, T.; Li, C.; Liu, P. One-Pot Two-Step Strategy for Efficient Synthesis of 3-Aryl-4-(arylthio)-1H-pyrazol-5-amines Derivatives. Chinese Journal of Organic Chemistry 2022, 42, 226. doi:10.6023/cjoc202107045
• He, Z.; Charleton, C.; Devine, R.; Kelada, M.; Walsh, J. M.; Conway, G. E.; Gunes, S.; Mondala, J. R. M.; Tian, F.; Tiwari, B. K.; Kinsella, G. K.; Malone, R.; O'Shea, D.; Devereux, M.; Wang, W.; Cullen, P. J.; Stephens, J. C.; Curtin, J. F. Enhanced pyrazolopyrimidinones cytotoxicity against glioblastoma cells activated by ROS-Generating cold atmospheric plasma. European journal of medicinal chemistry 2021, 224, 113736. doi:10.1016/j.ejmech.2021.113736
• Kumar, H.; Das, R.; Choithramani, A.; Gupta, A.; Khude, D.; Bothra, G.; Shard, A. Efficient Green Protocols for the Preparation of Pyrazolopyrimidines. ChemistrySelect 2021, 6, 5807–5837. doi:10.1002/slct.202101298
• Wei, Y.; Liu, P.; Liu, Y.; He, J.; Li, X.; Li, S.; Zhao, J. NIS-promoted three-component reaction of 3-oxo-3-arylpropanenitriles with arylsulfonyl hydrazides. Organic & biomolecular chemistry 2021, 19, 3932–3939. doi:10.1039/d1ob00438g
• He, Z.; C, C.; Devine, R.; Kelada, M.; Walsh, J. M.; G, C.; Gunes, S.; Jrm, M.; Tian, F.; Tiwari, B. K.; Gk, K.; Malone, R.; D, O.; Devereux, M.; W, W.; Cullen, P. J.; Stephens, J. C.; Curtin, J. F. Synergistic Cytotoxicity Between Cold Atmospheric Plasma and Pyrazolopyrimidinones Against Glioblastoma Cells. Cold Spring Harbor Laboratory 2021. doi:10.1101/2021.02.04.429831
• Mekky, A. E. M.; Ahmed, M. S. M.; Sanad, S. M. H.; Abdallah, Z. A. Bis(benzofuran-enaminone) hybrid possessing piperazine linker: Versatile precursor for microwave assisted synthesis of bis(pyrido[2',3':3,4]pyrazolo[1,5-a]pyrimidines). Synthetic Communications 2021, 51, 1085–1099. doi:10.1080/00397911.2020.1867745
• Zhu, R.; Reddy, R.; Ding, M.; Xu, M.; Deng, C.; Tadayon, S.; Li, H.; Depew, K. M.; Lane, B. S. Development and Scale-Up of a Continuous Manufacturing Process for a Hydrazine Condensation Reaction. Organic Process Research & Development 2021, 25, 199–205. doi:10.1021/acs.oprd.0c00424
• Al-Azmi, A. Pyrazolo[1,5-a]pyrimidines: A Close Look into their Synthesis and Applications. Current Organic Chemistry 2019, 23, 721–743. doi:10.2174/1385272823666190410145238
• Hoang, G. L.; Streit, A. D.; Ellman, J. A. Three-Component Coupling of Aldehydes, Aminopyrazoles, and Sulfoxonium Ylides via Rhodium(III)-Catalyzed Imidoyl C-H Activation: Synthesis of Pyrazolo[1,5- a]pyrimidines. The Journal of organic chemistry 2018, 83, 15347–15360. doi:10.1021/acs.joc.8b02606
• He, Z. doi:10.21427/4661-1k23

Explore citations to this article at