Enantioselective phase-transfer catalyzed alkylation of 1-methyl-7-methoxy-2-tetralone: an effective route to dezocine

Ruipeng Li, Zhenren Liu, Liang Chen, Jing Pan and Weicheng Zhou

Beilstein J. Org. Chem. 2018, 14, 1421–1427. doi:10.3762/bjoc.14.119

Supporting Information

Supporting Information File 1: Synthesis of catalysts C1C17, synthesis of dezocine, 1H NMR and MS spectra of catalysts C1–C17 and chiral HPLC diagrams of 3. 1H NMR, 13C NMR, MS spectra of 3. 1H NMR, MS spectra HPLC diagrams of dezocine.
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