The mechanochemical synthesis of quinazolin-4(3H)-ones by controlling the reactivity of IBX

Scholarly Works

• Wang, L.; Zhang, Y.; Xu, H.; Zhang, Z. Mechanosynthesis of N-heterocyclic compounds via ball milling. Tetrahedron 2025, 185, 134842. doi:10.1016/j.tet.2025.134842
• Recent advances in the mechanochemical synthesis and derivatization of heterocycles. Advances in Heterocyclic Chemistry; Elsevier, 2025; pp 133–224. doi:10.1016/bs.aihch.2025.05.002
• Bera, S. K.; Behera, S.; De Luca, L.; Basoccu, F.; Mocci, R.; Porcheddu, A. Unveiling the Untapped Potential of Bertagnini's Salts in Microwave-Assisted Synthesis of Quinazolinones. Molecules (Basel, Switzerland) 2024, 29, 1986. doi:10.3390/molecules29091986
• Kumar, S.; Arora, A.; Singh, S. K.; Kumar, R.; Shankar, B.; Singh, B. K. Phenyliodine bis(trifluoroacetate) as a sustainable reagent: exploring its significance in organic synthesis. Organic & biomolecular chemistry 2024, 22, 3109–3185. doi:10.1039/d3ob01964k
• Varala, R.; Seema, V.; Alam, M. M.; Dubasi, N.; Vummadi, R. D. Iodoxybenzoic Acid (IBX) in Organic Synthesis: A Septennial Review. Current organic synthesis 2024, 21, 607–664. doi:10.2174/0115701794263252230924074035
• Hou, S.; Xu, J.; Wang, J.; Wang, H.; Zhang, P. Mechanochemical Oxidative Coupling of Amine to Azo-based Polymers by Hypervalent Iodine Oxidant. Chemistry (Weinheim an der Bergstrasse, Germany) 2023, 30, e202303126. doi:10.1002/chem.202303126
• Brandão, P.; Pineiro, M. doi:10.1002/9781119889878.ch11
• Oduselu, G. O.; Aderohunmu, D. V.; Ajani, O. O.; Elebiju, O. F.; Ogunnupebi, T. A.; Adebiyi, E. Synthesis, in silico and in vitro antimicrobial efficacy of substituted arylidene-based quinazolin-4(3H)-one motifs. Frontiers in chemistry 2023, 11, 1264824. doi:10.3389/fchem.2023.1264824
• Sihag, M.; Soni, R.; Rani, N.; Kinger, M.; Kumar Aneja, D. Recent Synthetic Applications of Hypervalent Iodine Reagents. A Review in Three Installments: Installment I. Organic Preparations and Procedures International 2022, 55, 1–62. doi:10.1080/00304948.2022.2113964
• Pan, L.; Zheng, L.; Chen, Y.; Ke, Z.; Yeung, Y. A Mechanochemical, Catalyst‐Free Cascade Synthesis of 1,3‐Diols and 1,4‐Iodoalcohols Using Styrenes and Hypervalent Iodine Reagents. Angewandte Chemie 2022, 134. doi:10.1002/ange.202207926
• Pan, L.; Zheng, L.; Chen, Y.; Ke, Z.; Yeung, Y.-Y. A Mechanochemical, Catalyst-Free Cascade Synthesis of 1,3-Diols and 1,4-Iodoalcohols Using Styrenes and Hypervalent Iodine Reagents. Angewandte Chemie (International ed. in English) 2022, 61, e202207926. doi:10.1002/anie.202207926
• Bera, S. K.; Bhanja, R.; Mal, P. DDQ in mechanochemical C-N coupling reactions. Beilstein journal of organic chemistry 2022, 18, 639–646. doi:10.3762/bjoc.18.64
• Parida, K. N.; Moorthy, J. N. Catalytic Oxidations with ortho-Substituted Modified IBXs. Synlett 2022, 34, 495–506. doi:10.1055/a-1813-7319
• Ardila-Fierro, K. J.; Hernández, J. G. Sustainability Assessment of Mechanochemistry by Using the Twelve Principles of Green Chemistry. ChemSusChem 2021, 14, 2145–2162. doi:10.1002/cssc.202100478
• Dayaker, G.; Tan, D.; Biggins, N.; Shelam, A.; Do, J.-L.; Katsenis, A. D.; Friščić, T. Catalytic Room-Temperature C−N Coupling of Amides and Isocyanates by Using Mechanochemistry. ChemSusChem 2020, 13, 2966–2972. doi:10.1002/cssc.201902576
• Bal, A.; Maiti, S.; Mal, P. Strategies to Control Hypervalent Iodine - Primary Amine Reactions. Chemistry, an Asian journal 2020, 15, 624–635. doi:10.1002/asia.201901683
• Halder, A.; Maiti, D.; De Sarkar, S. Mechanochemical Synthesis of Functionalized Quinolines by Iodine Mediated Oxidative Annulation. Chemistry, an Asian journal 2020, 15, 577–580. doi:10.1002/asia.201901758
• Maiti, S.; Kim, J.; Park, J.-H.; Nam, D.; Bin Lee, J.; Kim, Y.-J.; Kee, J.-M.; Seo, J. K.; Myung, K.; Rohde, J.-U.; Choe, W.; Kwon, O.-H.; Hong, S. Y. Chemoselective Trifluoroethylation Reactions of Quinazolinones and Identification of Photostability. The Journal of organic chemistry 2019, 84, 6737–6751. doi:10.1021/acs.joc.9b00470
• Choudhuri, K.; Maiti, S.; Mal, P. Iodine(III) Enabled Dehydrogenative Aryl C−S Coupling by in situ Generated Sulfenium Ion. Advanced Synthesis & Catalysis 2019, 361, 1092–1101. doi:10.1002/adsc.201801510

Explore citations to this article at