Hoveyda–Grubbs catalysts with an N→Ru coordinate bond in a six-membered ring. Synthesis of stable, industrially scalable, highly efficient ruthenium metathesis catalysts and 2-vinylbenzylamine ligands as their precursors

Kirill B. Polyanskii,
Kseniia A. Alekseeva,
Pavel V. Raspertov,
Pavel A. Kumandin,
Eugeniya V. Nikitina,
Atash V. Gurbanov and
Fedor I. Zubkov

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Beilstein J. Org. Chem. 2019, 15, 769–779, doi:10.3762/bjoc.15.73

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Solid-phase synthesis of biaryl bicyclic peptides containing a 3-aryltyrosine or a 4-arylphenylalanine moiety

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Àngel Oliveras,
Lidia Feliu and
Marta Planas

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Beilstein J. Org. Chem. 2019, 15, 761–768, doi:10.3762/bjoc.15.72

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Diastereo- and enantioselective preparation of cyclopropanol derivatives

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Beilstein J. Org. Chem. 2019, 15, 752–760, doi:10.3762/bjoc.15.71

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Beilstein J. Org. Chem. 2019, 15, 746–751, doi:10.3762/bjoc.15.70

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Synthesis of polydicyclopentadiene using the Cp₂TiCl₂/Et₂AlCl catalytic system and thin-layer oxidation of the polymer in air

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Ludmila S. Soroka,
Alex A. Lyapkov,
Мekhman S. Yusubov and
Francis Verpoort

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Beilstein J. Org. Chem. 2019, 15, 733–745, doi:10.3762/bjoc.15.69

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Synthesis of functionalized diazocines for application as building blocks in photo- and mechanoresponsive materials

Widukind Moormann,
Daniel Langbehn and
Rainer Herges

Full Research Paper
Published 20 Mar 2019

Beilstein J. Org. Chem. 2019, 15, 727–732, doi:10.3762/bjoc.15.68

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Efficient synthesis of 4-substituted-ortho-phthalaldehyde analogues: toward the emergence of new building blocks

Clémence Moitessier,
Ahmad Rifai,
Pierre-Edouard Danjou,
Isabelle Mallard and
Francine Cazier-Dennin

Full Research Paper
Published 19 Mar 2019

Beilstein J. Org. Chem. 2019, 15, 721–726, doi:10.3762/bjoc.15.67

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Homo- and hetero-difunctionalized β-cyclodextrins: Short direct synthesis in gram scale and analysis of regiochemistry

Gábor Benkovics,
Mihály Bálint,
Éva Fenyvesi,
Erzsébet Varga,
Szabolcs Béni,
Konstantina Yannakopoulou and
Milo Malanga

Full Research Paper
Published 18 Mar 2019

Beilstein J. Org. Chem. 2019, 15, 710–720, doi:10.3762/bjoc.15.66

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An efficient and concise access to 2-amino-4H-benzothiopyran-4-one derivatives

Peng Li,
Yongqi Wu,
Tingting Zhang,
Chen Ma,
Ziyun Lin,
Gang Li and
Haihong Huang

Full Research Paper
Published 18 Mar 2019

Beilstein J. Org. Chem. 2019, 15, 703–709, doi:10.3762/bjoc.15.65

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New sesquiterpenoids from the South China Sea soft corals Clavularia viridis and Lemnalia flava

Qihao Wu,
Yuan Gao,
Meng-Meng Zhang,
Li Sheng,
Jia Li,
Xu-Wen Li,
Hong Wang and
Yue-Wei Guo

Full Research Paper
Published 15 Mar 2019

Beilstein J. Org. Chem. 2019, 15, 695–702, doi:10.3762/bjoc.15.64

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Supporting Information File 1: Compound library structures and screening results.
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Supporting Information File 2: Full dose–response curves.
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Supporting Information File 3: Competition assay efficacy and potency data.
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Non-native autoinducer analogs capable of modulating the SdiA quorum sensing receptor in Salmonella enterica serovar Typhimurium

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Antibacterials, bacterial small molecule interactions and quorum sensing

Latest Articles

Hoveyda–Grubbs catalysts with an N→Ru coordinate bond in a six-membered ring. Synthesis of stable, industrially scalable, highly efficient ruthenium metathesis catalysts and 2-vinylbenzylamine ligands as their precursors

Solid-phase synthesis of biaryl bicyclic peptides containing a 3-aryltyrosine or a 4-arylphenylalanine moiety

Diastereo- and enantioselective preparation of cyclopropanol derivatives

Tuning the stability of alkoxyisopropyl protection groups

Synthesis of polydicyclopentadiene using the Cp₂TiCl₂/Et₂AlCl catalytic system and thin-layer oxidation of the polymer in air

Synthesis of functionalized diazocines for application as building blocks in photo- and mechanoresponsive materials

Efficient synthesis of 4-substituted-ortho-phthalaldehyde analogues: toward the emergence of new building blocks

Homo- and hetero-difunctionalized β-cyclodextrins: Short direct synthesis in gram scale and analysis of regiochemistry

An efficient and concise access to 2-amino-4H-benzothiopyran-4-one derivatives

New sesquiterpenoids from the South China Sea soft corals Clavularia viridis and Lemnalia flava

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