Efficient synthesis of dipeptide analogues of α-fluorinated β-aminophosphonates

Marcin Kaźmierczak and Henryk Koroniak
Beilstein J. Org. Chem. 2020, 16, 756–762. https://doi.org/10.3762/bjoc.16.69

Supporting Information

Supporting Information File 1: Optimization of reaction conditions data, characterization data, copies of NMR spectra for compounds 13–15, single crystal X-ray data for compound 14c.
Format: PDF Size: 5.7 MB Download
Supporting Information File 2: CIF file of 14c.
Format: CIF Size: 380.9 KB Download

Cite the Following Article

Efficient synthesis of dipeptide analogues of α-fluorinated β-aminophosphonates
Marcin Kaźmierczak and Henryk Koroniak
Beilstein J. Org. Chem. 2020, 16, 756–762. https://doi.org/10.3762/bjoc.16.69

How to Cite

Kaźmierczak, M.; Koroniak, H. Beilstein J. Org. Chem. 2020, 16, 756–762. doi:10.3762/bjoc.16.69

Download Citation

Citation data can be downloaded as file using the "Download" button or used for copy/paste from the text window below.
Citation data in RIS format can be imported by all major citation management software, including EndNote, ProCite, RefWorks, and Zotero.

Presentation Graphic

Picture with graphical abstract, title and authors for social media postings and presentations.
Format: PNG Size: 104.4 KB Download

Citations to This Article

Up to 20 of the most recent references are displayed here.

Scholarly Works

  • Wątroba, K.; Pawełczak, M.; Kaźmierczak, M. Dipeptide analogues of fluorinated aminophosphonic acid sodium salts as moderate competitive inhibitors of cathepsin C. Beilstein journal of organic chemistry 2023, 19, 434–439. doi:10.3762/bjoc.19.33
  • Bilska-Markowska, M.; Kaźmierczak, M. Horner-Wadsworth-Emmons reaction as an excellent tool in the synthesis of fluoro-containing biologically important compounds. Organic & biomolecular chemistry 2023, 21, 1095–1120. doi:10.1039/d2ob01969h
  • Bilska-Markowska, M.; Jankowski, W.; Hoffmann, M.; Kaźmierczak, M. Design and Synthesis of New α-hydroxy β-fluoro/β-trifluoromethyl and Unsaturated Phosphonates from Carbohydrate-Derived Building Blocks via Pudovik and Horner-Wadsworth-Emmons Reactions. Molecules (Basel, Switzerland) 2022, 27, 5404. doi:10.3390/molecules27175404
  • Kaźmierczak, M.; Dutkiewicz, G.; Koroniak, H. Deoxyfluorinating reagents as tools for γ-amino-α-hydroxyphosphonate modification. Organic & biomolecular chemistry 2022, 20, 5615–5623. doi:10.1039/d2ob00915c
  • Kaźmierczak, M.; Siodła, T.; Koroniak, H. Stereoselective synthesis and investigation of mechanism of trifluoromethylated cyclopropylphosphonate. Journal of Fluorine Chemistry 2022, 254, 109934. doi:10.1016/j.jfluchem.2021.109934
  • Bilska‐Markowska, M.; Patyk‐Kaźmierczak, E.; Lusina, A. Synthesis of Fluorinated Amides Starting from Carbohydrates Based on the Claisen Rearrangement. European Journal of Organic Chemistry 2022, 2022. doi:10.1002/ejoc.202101378
  • Kaźmierczak, M.; Bilska-Markowska, M. Diethylaminosulfur Trifluoride (DAST) Mediated Transformations Leading to Valuable Building Blocks and Bioactive Compounds. European Journal of Organic Chemistry 2021, 2021, 5585–5604. doi:10.1002/ejoc.202101027
  • Kaźmierczak, M.; Dutkiewicz, G.; Cytlak, T. Application of α-Amino-β-fluorophosphonates in Construction of their Dipeptide Analogues. Synthesis 2020, 52, 2364–2372. doi:10.1055/s-0040-1707813
Other Beilstein-Institut Open Science Activities