Synthesis of 1-indolyl-3,5,8-substituted γ-carbolines: one-pot solvent-free protocol and biological evaluation

Premansh Dudhe, Mena Asha Krishnan, Kratika Yadav, Diptendu Roy, Krishnan Venkatasubbaiah, Biswarup Pathak and Venkatesh Chelvam

Beilstein J. Org. Chem. 2021, 17, 1453–1463. doi:10.3762/bjoc.17.101

Supporting Information

Supporting Information File 1: Copies of 1H, 13C NMR spectra of 1a–h, 3aa–ac, 3ba–bc, 3da, 3ea, 3ga, 12a–b, 12e–f, 12i, 14d, 14g and 15, UV calibration curves in different organic solvents for γ-carboline 3ac, and single-crystal XRD data of 3ac.
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