α,β-Aziridinylphosphonates by lithium amide-induced phosphonyl migration from nitrogen to carbon in terminal aziridines

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• Korb, M.; Lehrich, S. W.; Lang, H. Reactivity of Ferrocenyl Phosphates Bearing (Hetero-)Aromatics and [3]Ferrocenophanes toward Anionic Phospho-Fries Rearrangements. The Journal of organic chemistry 2017, 82, 3102–3124. doi:10.1021/acs.joc.7b00030
• Dogan, Ö.; Cakir, S. P.; Beksultanova, N.; Altanlar, N.; Şimşek, D.; Karabıyık, H. Enantioselective synthesis of new chiral 2-aziridinyl phosphonates and studies of their biological activities. Tetrahedron: Asymmetry 2017, 28, 324–329. doi:10.1016/j.tetasy.2017.01.003
• Parisi, G.; Capitanelli, E.; Pierro, A.; Romanazzi, G.; Clarkson, G. J.; Degennaro, L.; Luisi, R. Easy access to constrained peptidomimetics and 2,2-disubstituted azetidines by the unexpected reactivity profile of α-lithiated N-Boc-azetidines. Chemical communications (Cambridge, England) 2015, 51, 15588–15591. doi:10.1039/c5cc06323j
• Kadina, A. P.; Kashemirov, B. A.; Oertell, K.; Batra, V. K.; Wilson, S. H.; Goodman, M. F.; McKenna, C. E. Two Scaffolds from Two Flips: (α,β)/(β,γ) CH2/NH "Met-Im" Analogues of dTTP. Organic letters 2015, 17, 2586–2589. doi:10.1021/acs.orglett.5b00799
• Ordóñez, M.; Viveros-Ceballos, J. L.; Cativiela, C.; Sayago, F. J. An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives. Tetrahedron 2015, 71, 1745–1784. doi:10.1016/j.tet.2015.01.029
• Tao, J.; Jin, L.-M.; Zhang, X. P. Synthesis of chiral N-phosphoryl aziridines through enantioselective aziridination of alkenes with phosphoryl azide via Co(II)-based metalloradical catalysis. Beilstein journal of organic chemistry 2014, 10, 1282–1289. doi:10.3762/bjoc.10.129
• Strumfs, B.; Hermane, J.; Belyakov, S.; Trapencieris, P. Acyl migration from N to C in aziridine-2-carboxylic esters. Tetrahedron 2014, 70, 355–362. doi:10.1016/j.tet.2013.11.052
• Kurhade, S.; Ramaiah, P. A.; Prathipati, P.; Bhuniya, D. Unprecedented N→C[1,4] Boc migration: synthesis of 3-carboxyl functionalized 7-azaindolo[2,1-c][1,4]benzoxazine ring system. Tetrahedron 2013, 69, 1354–1362. doi:10.1016/j.tet.2012.11.073
• Keniche, A.; Mezrai, A.; Mulengi, J. K. Synthesis of a Novel Class of Phosphonoaziridines as Interesting Antibacterial Agents. The Open Conference Proceedings Journal 2011, 2, 28–35. doi:10.2174/2210289201102010028
• Dogan, Ö.; Babiz, H.; Gozen, A. G.; Budak, S. Synthesis of 2-aziridinyl phosphonates by modified Gabriel-Cromwell reaction and their antibacterial activities. European journal of medicinal chemistry 2011, 46, 2485–2489. doi:10.1016/j.ejmech.2011.03.037

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