Supporting Information
| Supporting Information File 1: General experimental conditions, experimental procedures and data, copies of 1H NMR and 13C NMR spectra for compounds 3, syn-5, 8, and 10–13. | ||
| Format: PDF | Size: 1.6 MB | Download |
| Supporting Information File 2: CIF-file of compound syn-5b. | ||
| Format: CIF | Size: 21.7 KB | Download |
Cite the Following Article
Asymmetric synthesis of γ-chloro-α,β-diamino- and β,γ-aziridino-α-aminoacylpyrrolidines and -piperidines via stereoselective Mannich-type additions of N-(diphenylmethylene)glycinamides across α-chloro-N-sulfinylimines
Gert Callebaut, Sven Mangelinckx, Pieter Van der Veken, Karl W. Törnroos, Koen Augustyns and Norbert De Kimpe
Beilstein J. Org. Chem. 2012, 8, 2124–2131.
https://doi.org/10.3762/bjoc.8.239
How to Cite
Callebaut, G.; Mangelinckx, S.; Van der Veken, P.; Törnroos, K. W.; Augustyns, K.; De Kimpe, N. Beilstein J. Org. Chem. 2012, 8, 2124–2131. doi:10.3762/bjoc.8.239
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- Wu, G.; Wang, J.; Liu, C.; Sun, M.; Zhang, L.; Ma, Y.; Cheng, R.; Ye, J. Transition metal-free, visible-light-mediated construction of α,β-diamino esters via decarboxylative radical addition at room temperature. Organic Chemistry Frontiers 2019, 6, 2245–2249. doi:10.1039/c9qo00407f
- Zhang, H.; Yang, Z.; Zhao, B. N.; Li, G. Group-Assisted Purification Chemistry for Asymmetric Mannich-type Reaction of Chiral N-Phosphonyl Imines with Azlactones Leading to Syntheses of α-Quaternary α,β-Diamino Acid Derivatives †. The Journal of organic chemistry 2017, 83, 644–655. doi:10.1021/acs.joc.7b02556
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- Guerola, M.; Sánchez-Roselló, M.; Mulet, C.; del Pozo, C.; Fustero, S. Asymmetric intramolecular aza-Michael reaction in desymmetrization processes. Total synthesis of hippodamine and epi-hippodamine. Organic letters 2015, 17, 960–963. doi:10.1021/acs.orglett.5b00054
- Pellissier, H. Recent Developments in Asymmetric Aziridination. Advanced Synthesis & Catalysis 2014, 356, 1899–1935. doi:10.1002/adsc.201400312
- Callebaut, G.; Meiresonne, T.; De Kimpe, N.; Mangelinckx, S. Synthesis and reactivity of 2-(carboxymethyl)aziridine derivatives. Chemical reviews 2014, 114, 7954–8015. doi:10.1021/cr400582d
- Callebaut, G.; Colpaert, F.; Nonn, M.; Kiss, L.; Sillanpää, R.; Törnroos, K. W.; Fülöp, F.; De Kimpe, N.; Mangelinckx, S. Asymmetric synthesis of chloroisothreonine derivatives via syn-stereoselective Mannich-type additions across N-sulfinyl-α-chloroimines. Organic & biomolecular chemistry 2014, 12, 3393–3405. doi:10.1039/c4ob00243a
- Kattamuri, P. V.; Xiong, Y.; Pan, Y.; Li, G. N,N-DIIsopropyl-N-phosphonyl imines lead to efficient asymmetric synthesis of aziridine-2-carboxylic esters. Organic & biomolecular chemistry 2013, 11, 3400–3408. doi:10.1039/c3ob40251g
- Callebaut, G. Ph.D. Thesis, Jan 1, 2013.
