Synthesis of new dihydroberberine and tetrahydroberberine analogues and evaluation of their antiproliferative activity on NCI-H1975 cells

Giacomo Mari,
Lucia De Crescentini,
Serena Benedetti,
Francesco Palma,
Stefania Santeusanio and
Fabio Mantellini

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Beilstein J. Org. Chem. 2020, 16, 1606–1616, doi:10.3762/bjoc.16.133

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Antibacterial scalarane from Doriprismatica stellata nudibranchs (Gastropoda, Nudibranchia), egg ribbons, and their dietary sponge Spongia cf. agaricina (Demospongiae, Dictyoceratida)

Cora Hertzer,
Stefan Kehraus,
Nils Böhringer,
Fontje Kaligis,
Robert Bara,
Dirk Erpenbeck,
Gert Wörheide,
Till F. Schäberle,
Heike Wägele and
Gabriele M. König

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Beilstein J. Org. Chem. 2020, 16, 1596–1605, doi:10.3762/bjoc.16.132

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A dynamic combinatorial library for biomimetic recognition of dipeptides in water

Florian Klepel and
Bart Jan Ravoo

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Beilstein J. Org. Chem. 2020, 16, 1588–1595, doi:10.3762/bjoc.16.131

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Azidophosphonium salt-directed chemoselective synthesis of (E)/(Z)-cinnamyl-1H-triazoles and regiospecific access to bromomethylcoumarins from Morita–Baylis–Hillman adducts

Soundararajan Karthikeyan,
Radha Krishnan Shobana,
Kamarajapurathu Raju Subimol,
J. Helen Ratna Monica and
Ayyanoth Karthik Krishna Kumar

Full Research Paper
Published 01 Jul 2020

Beilstein J. Org. Chem. 2020, 16, 1579–1587, doi:10.3762/bjoc.16.130

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NHC-catalyzed enantioselective synthesis of β-trifluoromethyl-β-hydroxyamides

Alyn T. Davies,
Mark D. Greenhalgh,
Alexandra M. Z. Slawin and
Andrew D. Smith

Letter
Published 30 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1572–1578, doi:10.3762/bjoc.16.129

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Five-component, one-pot synthesis of an electroactive rotaxane comprising a bisferrocene macrocycle

Natalie Lagesse,
Luca Pisciottani,
Maxime Douarre,
Pascale Godard,
Brice Kauffmann,
Vicente Martí-Centelles and
Nathan D. McClenaghan

Full Research Paper
Published 30 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1564–1571, doi:10.3762/bjoc.16.128

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Mechanochemical green synthesis of hyper-crosslinked cyclodextrin polymers

Alberto Rubin Pedrazzo,
Fabrizio Caldera,
Marco Zanetti,
Silvia Lucia Appleton,
Nilesh Kumar Dhakar and
Francesco Trotta

Full Research Paper
Published 29 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1554–1563, doi:10.3762/bjoc.16.127

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Photoredox-catalyzed silyldifluoromethylation of silyl enol ethers

Vyacheslav I. Supranovich,
Vitalij V. Levin and
Alexander D. Dilman

Letter
Published 29 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1550–1553, doi:10.3762/bjoc.16.126

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Heterogeneous photocatalysis in flow chemical reactors

Christopher G. Thomson,
Ai-Lan Lee and
Filipe Vilela

Review
Published 26 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1495–1549, doi:10.3762/bjoc.16.125

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4-Hydroxy-3-methyl-2(1H)-quinolone, originally discovered from a Brassicaceae plant, produced by a soil bacterium of the genus Burkholderia sp.: determination of a preferred tautomer and antioxidant activity

Dandan Li,
Naoya Oku,
Yukiko Shinozaki,
Yoichi Kurokawa and
Yasuhiro Igarashi

Letter
Published 26 Jun 2020

Beilstein J. Org. Chem. 2020, 16, 1489–1494, doi:10.3762/bjoc.16.124

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Supporting Information File 1: Experimental procedures and characterization data for new compounds. In addition, confirmatory crystallographic data are included.
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Organocatalytic asymmetric selenofunctionalization of tryptamine for the synthesis of hexahydropyrrolo[2,3-b]indole derivatives

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Transition-metal and organocatalysis in natural product synthesis

Latest Articles

Synthesis of new dihydroberberine and tetrahydroberberine analogues and evaluation of their antiproliferative activity on NCI-H1975 cells

Antibacterial scalarane from Doriprismatica stellata nudibranchs (Gastropoda, Nudibranchia), egg ribbons, and their dietary sponge Spongia cf. agaricina (Demospongiae, Dictyoceratida)

A dynamic combinatorial library for biomimetic recognition of dipeptides in water

Azidophosphonium salt-directed chemoselective synthesis of (E)/(Z)-cinnamyl-1H-triazoles and regiospecific access to bromomethylcoumarins from Morita–Baylis–Hillman adducts

NHC-catalyzed enantioselective synthesis of β-trifluoromethyl-β-hydroxyamides

Five-component, one-pot synthesis of an electroactive rotaxane comprising a bisferrocene macrocycle

Mechanochemical green synthesis of hyper-crosslinked cyclodextrin polymers

Photoredox-catalyzed silyldifluoromethylation of silyl enol ethers

Heterogeneous photocatalysis in flow chemical reactors

4-Hydroxy-3-methyl-2(1H)-quinolone, originally discovered from a Brassicaceae plant, produced by a soil bacterium of the genus Burkholderia sp.: determination of a preferred tautomer and antioxidant activity

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