2 article(s) from Abbiati, Giorgio
Examples of drugs embodying unnatural amino acids.
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Examples of biologically active compounds embodying constrained analogues of tryptophan.
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Planned Diels–Alder reactions for the synthesis of tetrahydrocarbazoles as constrained analogues of...
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Structure elucidation of diastereoisomeric tetrahydrocarbazoles 3a and 3’a via NMR experiments.
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Synthesis of unprotected tryptophan derivatives 6a–e.
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Plausible reaction mechanism for the cycloaddition reactions of indoles 1a–h with 2 in toluene.
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Cycloaddition reaction of 2-vinylindole 1k and methyl 2-acetamidoacrylate (2).
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Beilstein J. Org. Chem. 2015, 11, 1997–2006, doi:10.3762/bjoc.11.216
General reaction mechanism for Ag(I)-catalyzed A3-coupling reactions.
A3-coupling reaction catalyzed by polystyrene-supported NHC–silver halides.
Various NHC–Ag(I) complexes used as catalysts for A3-coupling.
Proposed reaction mechanism for NHC–AgCl catalyzed A3-coupling reactions.
Liu’s synthesis of pyrrole-2-carboxaldehydes 4.
Proposed reaction mechanism for Liu’s synthesis of pyrrole-2-carboxaldehydes 4.
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Gold-catalyzed synthesis of propargylamines 1.
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A3-coupling catalyzed by phosphinamidic Au(III) metallacycle 6.
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A3-coupling applied to aldehyde-containing oligosaccharides 8.
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A3-MCR for the preparation of propargylamine-substituted indoles 9.
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A3-coupling interceded synthesis of furans 12.
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A3/KA2-coupling mediated synthesis of functionalized dihydropyrazoles 13 and polycyclic dihydropyra...
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Au(I)-catalyzed entry to cyclic carbamimidates 17 via an A3-coupling-type approach.
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Proposed reaction mechanism for the Au(I)-catalyzed synthesis of cyclic carbamimidates 17.
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Chiral trans-1-diphenylphosphino-2-aminocyclohexane–Au(I) complex 20.
A3-coupling-type synthesis of oxazoles 21 catalyzed by Au(III)–salen complex.
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Proposed reaction mechanism for the synthesis of oxazoles 21.
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Synthesis of propargyl ethyl ethers 24 by an A3-coupling-type reaction.
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General mechanism of Ag(I)-catalyzed MCRs of 2-alkynylbenzaldehydes, amines and nucleophiles.
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General synthetic pathway to 1,3-disubstituted-1,2-dihydroisoquinolines.
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Synthesis of 1,3-disubstituted-1,2-dihydroisoquinolines 29.
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Synthesis of 1,3-disubstituted-1,2-dihydroisoquinolines 35 and 36.
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Rh(II)/Ag(I) co-catalyzed synthesis of 1,3-disubstituted-1,2-dihydroisoquinolines 40.
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General synthetic pathway to 2-amino-1,2-dihydroquinolines.
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Synthesis of 2-amino-1,2-dihydroquinolines 47.
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Synthesis of tricyclic H-pyrazolo[5,1-a]isoquinoline 48.
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Synthesis of tricyclic H-pyrazolo[5,1-a]isoquinolines 48.
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Cu(II)/Ag(I) catalyzed synthesis of H-pyrazolo[5,1-a]isoquinolines 48.
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Synthesis of 2-aminopyrazolo[5,1-a]isoquinolines 53.
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Synthesis of 1-(isoquinolin-1-yl)guanidines 55.
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Ag(I)/Cu(I) catalyzed synthesis of 2-amino-H-pyrazolo[5,1-a]isoquinolines 58.
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Ag(I)/Ni(II) co-catalyzed synthesis of 3,4-dihydro-1H-pyridazino[6,1-a]isoquinoline-1,1-dicarboxyla...
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Ag(I) promoted activation of the α-carbon atom of the isocyanide group.
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Synthesis of dihydroimidazoles 65.
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Synthesis of oxazoles 68.
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Stereoselective synthesis of chiral butenolides 71.
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Proposed reaction mechanism for the synthesis of butenolides 71.
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Stereoselective three-component approach to pirrolidines 77 by means of a chiral auxiliary.
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Stereoselective three-component approach to pyrrolidines 81 and 82 by means of a chiral catalyst.
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Synthesis of substituted five-membered carbocyles 86.
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Synthesis of regioisomeric arylnaphthalene lactones.
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Enantioselective synthesis of spiroacetals 96 by Fañanás and Rodríguez .
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Enantioselective synthesis of spiroacetals 101 by Gong .
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Synthesis of polyfunctionalized fused bicyclic ketals 103 and bridged tricyclic ketals 104.
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Proposed reaction mechanism for the synthesis of ketals 103 and 104.
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Synthesis of β-alkoxyketones 108.
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Synthesis of N-methyl-1,4-dihydropyridines 112.
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Synthesis of tetrahydrocarbazoles 115–117.
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Plausible reaction mechanism for the synthesis of tetrahydrocarbazoles 115–117.
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Carboamination, carboalkoxylation and carbolactonization of terminal alkenes.
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Oxyarylation of alkenes with arylboronic acids and Selectfluor as reoxidant.
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Proposed reaction mechanism for oxyarylation of alkenes.
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Oxyarylation of alkenes with arylsilanes and Selectfluor as reoxidant.
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Oxyarylation of alkenes with arylsilanes and IBA as reoxidant.
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Beilstein J. Org. Chem. 2014, 10, 481–513, doi:10.3762/bjoc.10.46
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