This search combines search strings from the content search (i.e. "Full Text", "Author", "Title", "Abstract", or "Keywords") with "Article Type" and "Publication Date Range" using the AND operator.
Beilstein J. Org. Chem. 2014, 10, 369–383, doi:10.3762/bjoc.10.35
Natural products and other bioactive piperidine derivatives of type B.
Retrosynthetic analysis of piperidines B (X = OH or leaving group, PG = protecting group).
Synthesis of the protected amino acids 2. (a) KOH for 1b. b) PG–X = Cbz–Cl (1a–c), Boc2O (1d).
Synthesis of hydroxy ketones 7 (R = Me (a), Bn (b), Ph (c) and EtSMe (d); PG = Cbz (a–c), Boc (d)).
Synthesis of amides 5e and 5f and ketone 7e.
Synthesis of amino alcohols syn-9a–d and oxazolidinone 10a. (for 7a–c conditions A: H2 (1 atm), Pd/...
Competition between the Michaelis–Arbuzow process and the desired cyclodehydration of amino alcohol...
Initial synthesis of the trans-piperidinol 11a in diminished enantiopurity. aThe amino alcohol 9a o...
Synthesis of trans-piperidinol 11a in excellent ee.
Synthesis of L-733,060·HCl.