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Cite the Following Article
Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists
Constantinos G. Neochoritis, Maryam Kazemi Miraki, Eman M. M. Abdelraheem, Ewa Surmiak, Tryfon Zarganes-Tzitzikas, Beata Łabuzek, Tad A. Holak and Alexander Dömling
Beilstein J. Org. Chem. 2019, 15, 513–520.
https://doi.org/10.3762/bjoc.15.45
How to Cite
Neochoritis, C. G.; Kazemi Miraki, M.; Abdelraheem, E. M. M.; Surmiak, E.; Zarganes-Tzitzikas, T.; Łabuzek, B.; Holak, T. A.; Dömling, A. Beilstein J. Org. Chem. 2019, 15, 513–520. doi:10.3762/bjoc.15.45
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- Mohammadi Ziarani, G.; Hasani, S.; Mohajer, F.; Varma, R. S.; Rafiee, F. The Molecular Diversity of 1H-Indole-3-Carbaldehyde Derivatives and Their Role in Multicomponent Reactions. Topics in current chemistry (Cham) 2022, 380, 24. doi:10.1007/s41061-022-00379-5
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Patents
- ARONICA PIETRO; BROWN CHRISTOPER J; FERRER FERNANDO J; JOHANNES CHARLES W; KANNAN SRINIVASARAGHAVAN; LANE DAVID P; PARTRIDGE ANTHONY W; TAN YAW SING; VERMA CHANDRA S; YUEN TSZ YING. P53 ACTIVATOR PEPTIDOMIMETIC MACROCYCLES. EP 3986438 B1, April 16, 2025.
- DURDAĞI SERDAR; AVŞAR TIMUÇIN; ORHAN MÜGE DIDEM; PAKSOY MAIDE NUR; AYDIN GÜLŞAH; YURTSEVER MINE. DRG-MDM2-4 FOR USE AS A NOVEL MOUSE DOUBLE MINUTE 2 (MDM2) INHIBITOR. WO 2021167573 A1, Aug 26, 2021.
- ARONICA PIETRO; BROWN CHRISTOPER; FERRER FERNANDO; JOHANNES CHARLES; KANNAN SRINIVASARAGHAVAN; LANE DAVID; PARTRIDGE ANTHONY; TAN YAW SING; VERMA CHANDRA; YUEN TSZ YING. P53 ACTIVATOR PEPTIDOMIMETIC MACROCYCLES. WO 2020257153 A1, Dec 24, 2020.
- ARONICA PIETRO; BROWN CHRISTOPER; FERRER FERNANDO; JOHANNES CHARLES; KANNAN SRINIVASARAGHAVAN; LANE DAVID; PARTRIDGE ANTHONY; TAN YAW SING; VERMA CHANDRA; YUEN TSZ YING. P53 ACTIVATOR PEPTIDOMIMETIC MACROCYCLES. WO 2020257133 A1, Dec 24, 2020.
