3 article(s) from Budisa, Nediljko
A. Dependence of the lipophilicity (logP) on the number of fluorine atoms in a partially fluorinate...
Jump to Figure 1
Synthesis of the model compounds.
Jump to Scheme 1
Kinetics of the C-terminal ester hydrolysis.
Jump to Figure 2
Partitioning of the esters 1–5 between octan-1-ol and water. Insert: comparison with the other part...
Jump to Figure 3
Amide isomerism in the N-acetylprolyl fragment.
Jump to Scheme 2
Enhancement of the trans/cis thermodynamic preferences in the ester models as a function of the sol...
Jump to Figure 4
A. Four-state conformational equilibrium model used by Siebler et al.  for explanations of the elev...
Jump to Scheme 3
Elevation of the trans/cis ratio in derivatives of N-acyl proline may result from the enhanced n→π*...
Jump to Scheme 4
Synthesis of the model peptides.
Jump to Scheme 5
Mean residue molar circular dichroism (Δε) of peptides 8–10 in methanol (left) and aqueous phosphat...
Jump to Figure 5
Conformational analysis of the peptides by 1H DOSY NMR (D2O, 298 K). The theoretical values were ca...
Jump to Figure 6
Hydrolysis of the C-terminal 2,2-difluoroethyl esters of the oligopeptides in buffered deuterium ox...
Jump to Figure 7
Beilstein J. Org. Chem. 2017, 13, 2442–2457, doi:10.3762/bjoc.13.241
s-cis–s-trans Amide bond isomerism in an N-acyl-proline fragment.
Amino acids that have been compared in this study.
X-ray crystal structures of compounds 5–9. Carbon- grey, nitrogen – blue, oxygen – red, fluorine – ...
The relationship between the pKa of the ammonium function in the amino acid and the amide rotationa...
The double bond between C3 and C4 atoms in 3,4-dehydroproline residues induces an increase in the a...
Beilstein J. Org. Chem. 2016, 12, 589–593, doi:10.3762/bjoc.12.57
Protein design and dual-functionalization of TTL: periodate cleavage, oxime ligation and CuAAC.
Dual-functionalization of TTL: A) MALDI–MS spectra (red: modified protein (as marked below); black:...
SPR measurements: A) set-up showing different binding events of the double-functionalized TTL to EC...
Beilstein J. Org. Chem. 2015, 11, 784–791, doi:10.3762/bjoc.11.88
Subscribe to our Latest Articles RSS Feed.
Register and get informed about new articles.
Follow the Beilstein-Institut