2 article(s) from Suresh, Rajendran
Examples of biologically active oxazole and aminothiazole scaffolds.
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Strategies for the synthesis of 2,4,5-trisubstituted oxazole from azirine. a) I2, PPh3; b) NaH, 1H-...
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Scope of the α-azidochalcones. The reactions were carried out at reflux temperature, using 1 (1 mmo...
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Large-scale synthesis of 3i.
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Large-scale synthesis of 3i. a) At the start of the reaction, b) after the reaction.
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Acetyl derivative of 3d.
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ORTEP diagram of compound 5.
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Synthesis of S-methyl/benzylated products 6 and 7.
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Plausible mechanism proposed for the formation of 2,4,5-trisubstituted oxazoles 3.
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Reaction of vinyl azide 1 and 3 with ferric nitrate. Reactions were carried out at reflux temperatu...
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X-ray crystal structure of 4h.
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Beilstein J. Org. Chem. 2020, 16, 2108–2118, doi:10.3762/bjoc.16.178
Formation of substituted aziridine.
Various strategies for the formation of 2H-azirine.
Attempted reaction for the synthesis of 3a.
Synthesis of α-amido-1,3-diketone (3a–o). Reaction conditions: α-azidochalcone 1 (1.0 equiv) and ca...
Attempted reaction with acid derivatives.
Oxazole formation from 3.
Possible isomers for 7.
Synthesis of highly substituted 2-(trifluoromethyl)oxazoles (8a–e). Reaction conditions: α-azidocha...
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Mechanism for the formation of 8.
Beilstein J. Org. Chem. 2015, 11, 2021–2028, doi:10.3762/bjoc.11.219
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