Novel amide-functionalized chloramphenicol base bifunctional organocatalysts for enantioselective alcoholysis of meso-cyclic anhydrides
- Lingjun Xu,
- Shuwen Han,
- Linjie Yan,
- Haifeng Wang,
- Haihui Peng and
- Fener Chen
Beilstein J. Org. Chem. 2018, 14, 309–317, doi:10.3762/bjoc.14.19
Continuous-flow retro-Diels–Alder reaction: an efficient method for the preparation of pyrimidinone derivatives
- Imane Nekkaa,
- Márta Palkó,
- István M. Mándity and
- Ferenc Fülöp
Beilstein J. Org. Chem. 2018, 14, 318–324, doi:10.3762/bjoc.14.20
Recent developments in the asymmetric Reformatsky-type reaction
- Hélène Pellissier
Beilstein J. Org. Chem. 2018, 14, 325–344, doi:10.3762/bjoc.14.21
One-pot preparation of 4-aryl-3-bromocoumarins from 4-aryl-2-propynoic acids with diaryliodonium salts, TBAB, and Na2S2O8
- Teppei Sasaki,
- Katsuhiko Moriyama and
- Hideo Togo
Beilstein J. Org. Chem. 2018, 14, 345–353, doi:10.3762/bjoc.14.22
Diels–Alder cycloadditions of N-arylpyrroles via aryne intermediates using diaryliodonium salts
- Huangguan Chen,
- Jianwei Han and
- Limin Wang
Beilstein J. Org. Chem. 2018, 14, 354–363, doi:10.3762/bjoc.14.23
Synthesis of fluoro-functionalized diaryl-λ3-iodonium salts and their cytotoxicity against human lymphoma U937 cells
- Prajwalita Das,
- Etsuko Tokunaga,
- Hidehiko Akiyama,
- Hiroki Doi,
- Norimichi Saito and
- Norio Shibata
Beilstein J. Org. Chem. 2018, 14, 364–372, doi:10.3762/bjoc.14.24
Syn-selective silicon Mukaiyama-type aldol reactions of (pentafluoro-λ6-sulfanyl)acetic acid esters with aldehydes
- Anna-Lena Dreier,
- Andrej V. Matsnev,
- Joseph S. Thrasher and
- Günter Haufe
Beilstein J. Org. Chem. 2018, 14, 373–380, doi:10.3762/bjoc.14.25
Terahertz spectroscopy of 2,4,6-trinitrotoluene molecular solids from first principles
- Ido Azuri,
- Anna Hirsch,
- Anthony M. Reilly,
- Alexandre Tkatchenko,
- Shai Kendler,
- Oded Hod and
- Leeor Kronik
Beilstein J. Org. Chem. 2018, 14, 381–388, doi:10.3762/bjoc.14.26
The selective electrochemical fluorination of S-alkyl benzothioate and its derivatives
- Shunsuke Kuribayashi,
- Tomoyuki Kurioka,
- Shinsuke Inagi,
- Ho-Jung Lu,
- Biing-Jiun Uang and
- Toshio Fuchigami
Beilstein J. Org. Chem. 2018, 14, 389–396, doi:10.3762/bjoc.14.27
Preparation of trinucleotide phosphoramidites as synthons for the synthesis of gene libraries
- Ruth Suchsland,
- Bettina Appel and
- Sabine Müller
Beilstein J. Org. Chem. 2018, 14, 397–406, doi:10.3762/bjoc.14.28
Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting
- Lizeth Bodero,
- Paula López Rivas,
- Barbara Korsak,
- Torsten Hechler,
- Andreas Pahl,
- Christoph Müller,
- Daniela Arosio,
- Luca Pignataro,
- Cesare Gennari and
- Umberto Piarulli
Beilstein J. Org. Chem. 2018, 14, 407–415, doi:10.3762/bjoc.14.29
Synthetic and semi-synthetic approaches to unprotected N-glycan oxazolines
- Antony J. Fairbanks
Beilstein J. Org. Chem. 2018, 14, 416–429, doi:10.3762/bjoc.14.30
Palladium-catalyzed ortho-halogenations of acetanilides with N-halosuccinimides via direct sp2 C–H bond activation in ball mills
- Zi Liu,
- Hui Xu and
- Guan-Wu Wang
Beilstein J. Org. Chem. 2018, 14, 430–435, doi:10.3762/bjoc.14.31
Stimuli-responsive oligonucleotides in prodrug-based approaches for gene silencing
- Françoise Debart,
- Christelle Dupouy and
- Jean-Jacques Vasseur
Beilstein J. Org. Chem. 2018, 14, 436–469, doi:10.3762/bjoc.14.32
Latest development in the synthesis of ursodeoxycholic acid (UDCA): a critical review
- Fabio Tonin and
- Isabel W. C. E. Arends
Beilstein J. Org. Chem. 2018, 14, 470–483, doi:10.3762/bjoc.14.33
Carbohydrate inhibitors of cholera toxin
- Vajinder Kumar and
- W. Bruce Turnbull
Beilstein J. Org. Chem. 2018, 14, 484–498, doi:10.3762/bjoc.14.34
Functionalization of N-arylglycine esters: electrocatalytic access to C–C bonds mediated by n-Bu4NI
- Mi-Hai Luo,
- Yang-Ye Jiang,
- Kun Xu,
- Yong-Guo Liu,
- Bao-Guo Sun and
- Cheng-Chu Zeng
Beilstein J. Org. Chem. 2018, 14, 499–505, doi:10.3762/bjoc.14.35
Continuous multistep synthesis of 2-(azidomethyl)oxazoles
- Thaís A. Rossa,
- Nícolas S. Suveges,
- Marcus M. Sá,
- David Cantillo and
- C. Oliver Kappe
Beilstein J. Org. Chem. 2018, 14, 506–514, doi:10.3762/bjoc.14.36
Addition of dithi(ol)anylium tetrafluoroborates to α,β-unsaturated ketones
- Yu-Chieh Huang,
- An Nguyen,
- Simone Gräßle,
- Sylvia Vanderheiden,
- Nicole Jung and
- Stefan Bräse
Beilstein J. Org. Chem. 2018, 14, 515–522, doi:10.3762/bjoc.14.37
Synthesis and stability of strongly acidic benzamide derivatives
- Frederik Diness,
- Niels J. Bjerrum and
- Mikael Begtrup
Beilstein J. Org. Chem. 2018, 14, 523–530, doi:10.3762/bjoc.14.38
Oxidative cycloaddition of hydroxamic acids with dienes or guaiacols mediated by iodine(III) reagents
- Hisato Shimizu,
- Akira Yoshimura,
- Keiichi Noguchi,
- Victor N. Nemykin,
- Viktor V. Zhdankin and
- Akio Saito
Beilstein J. Org. Chem. 2018, 14, 531–536, doi:10.3762/bjoc.14.39
An alternative to hydrogenation processes. Electrocatalytic hydrogenation of benzophenone
- Cristina Mozo Mulero,
- Alfonso Sáez,
- Jesús Iniesta and
- Vicente Montiel
Beilstein J. Org. Chem. 2018, 14, 537–546, doi:10.3762/bjoc.14.40
Electrochemical Corey–Winter reaction. Reduction of thiocarbonates in aqueous methanol media and application to the synthesis of a naturally occurring α-pyrone
- Ernesto Emmanuel López-López,
- José Alvano Pérez-Bautista,
- Fernando Sartillo-Piscil and
- Bernardo A. Frontana-Uribe
Beilstein J. Org. Chem. 2018, 14, 547–552, doi:10.3762/bjoc.14.41
Investigations towards the stereoselective organocatalyzed Michael addition of dimethyl malonate to a racemic nitroalkene: possible route to the 4-methylpregabalin core structure
- Denisa Vargová,
- Rastislav Baran and
- Radovan Šebesta
Beilstein J. Org. Chem. 2018, 14, 553–559, doi:10.3762/bjoc.14.42
Mannich base-connected syntheses mediated by ortho-quinone methides
- Petra Barta,
- Ferenc Fülöp and
- István Szatmári
Beilstein J. Org. Chem. 2018, 14, 560–575, doi:10.3762/bjoc.14.43
Copper-catalyzed asymmetric methylation of fluoroalkylated pyruvates with dimethylzinc
- Kohsuke Aikawa,
- Kohei Yabuuchi,
- Kota Torii and
- Koichi Mikami
Beilstein J. Org. Chem. 2018, 14, 576–582, doi:10.3762/bjoc.14.44
High-yielding continuous-flow synthesis of antimalarial drug hydroxychloroquine
- Eric Yu,
- Hari P. R. Mangunuru,
- Nakul S. Telang,
- Caleb J. Kong,
- Jenson Verghese,
- Stanley E. Gilliland III,
- Saeed Ahmad,
- Raymond N. Dominey and
- B. Frank Gupton
Beilstein J. Org. Chem. 2018, 14, 583–592, doi:10.3762/bjoc.14.45
Diastereoselective auxiliary- and catalyst-controlled intramolecular aza-Michael reaction for the elaboration of enantioenriched 3-substituted isoindolinones. Application to the synthesis of a new pazinaclone analogue
- Romain Sallio,
- Stéphane Lebrun,
- Frédéric Capet,
- Francine Agbossou-Niedercorn,
- Christophe Michon and
- Eric Deniau
Beilstein J. Org. Chem. 2018, 14, 593–602, doi:10.3762/bjoc.14.46
