Nucleoside macrocycles formed by intramolecular click reaction: efficient cyclization of pyrimidine nucleosides decorated with 5'-azido residues and 5-octadiynyl side chains
- Jiang Liu,
- Peter Leonard,
- Sebastian L. Müller,
- Constantin Daniliuc and
- Frank Seela
Beilstein J. Org. Chem. 2018, 14, 2404–2410, doi:10.3762/bjoc.14.217
Synthesis of indolo[1,2-c]quinazolines from 2-alkynylaniline derivatives through Pd-catalyzed indole formation/cyclization with N,N-dimethylformamide dimethyl acetal
- Antonio Arcadi,
- Sandro Cacchi,
- Giancarlo Fabrizi,
- Francesca Ghirga,
- Antonella Goggiamani,
- Antonia Iazzetti and
- Fabio Marinelli
Beilstein J. Org. Chem. 2018, 14, 2411–2417, doi:10.3762/bjoc.14.218
Microfluidic light-driven synthesis of tetracyclic molecular architectures
- Javier Mateos,
- Nicholas Meneghini,
- Marcella Bonchio,
- Nadia Marino,
- Tommaso Carofiglio,
- Xavier Companyó and
- Luca Dell’Amico
Beilstein J. Org. Chem. 2018, 14, 2418–2424, doi:10.3762/bjoc.14.219
Efficient catalytic alkyne metathesis with a fluoroalkoxy-supported ditungsten(III) complex
- Henrike Ehrhorn,
- Janin Schlösser,
- Dirk Bockfeld and
- Matthias Tamm
Beilstein J. Org. Chem. 2018, 14, 2425–2434, doi:10.3762/bjoc.14.220
Cobalt- and rhodium-catalyzed carboxylation using carbon dioxide as the C1 source
- Tetsuaki Fujihara and
- Yasushi Tsuji
Beilstein J. Org. Chem. 2018, 14, 2435–2460, doi:10.3762/bjoc.14.221
Synthesis of eunicellane-type bicycles embedding a 1,3-cyclohexadiene moiety
- Alex Frichert,
- Peter G. Jones and
- Thomas Lindel
Beilstein J. Org. Chem. 2018, 14, 2461–2467, doi:10.3762/bjoc.14.222
Synergistic approach to polycycles through Suzuki–Miyaura cross coupling and metathesis as key steps
- Sambasivarao Kotha,
- Milind Meshram and
- Chandravathi Chakkapalli
Beilstein J. Org. Chem. 2018, 14, 2468–2481, doi:10.3762/bjoc.14.223
Synthesis of a leopolic acid-inspired tetramic acid with antimicrobial activity against multidrug-resistant bacteria
- Luce Mattio,
- Loana Musso,
- Leonardo Scaglioni,
- Andrea Pinto,
- Piera Anna Martino and
- Sabrina Dallavalle
Beilstein J. Org. Chem. 2018, 14, 2482–2487, doi:10.3762/bjoc.14.224
Calixazulenes: azulene-based calixarene analogues – an overview and recent supramolecular complexation studies
- Paris E. Georghiou,
- Shofiur Rahman,
- Abdullah Alodhayb,
- Hidetaka Nishimura,
- Jaehyun Lee,
- Atsushi Wakamiya and
- Lawrence T. Scott
Beilstein J. Org. Chem. 2018, 14, 2488–2494, doi:10.3762/bjoc.14.225
Comparative cell biological study of in vitro antitumor and antimetastatic activity on melanoma cells of GnRH-III-containing conjugates modified with short-chain fatty acids
- Eszter Lajkó,
- Sarah Spring,
- Rózsa Hegedüs,
- Beáta Biri-Kovács,
- Sven Ingebrandt,
- Gábor Mező and
- László Kőhidai
Beilstein J. Org. Chem. 2018, 14, 2495–2509, doi:10.3762/bjoc.14.226
Synthesis of dihydroquinazolines from 2-aminobenzylamine: N3-aryl derivatives with electron-withdrawing groups
- Nadia Gruber,
- Jimena E. Díaz and
- Liliana R. Orelli
Beilstein J. Org. Chem. 2018, 14, 2510–2519, doi:10.3762/bjoc.14.227
Synthesis of aryl sulfides via radical–radical cross coupling of electron-rich arenes using visible light photoredox catalysis
- Amrita Das,
- Mitasree Maity,
- Simon Malcherek,
- Burkhard König and
- Julia Rehbein
Beilstein J. Org. Chem. 2018, 14, 2520–2528, doi:10.3762/bjoc.14.228
Quinolines from the cyclocondensation of isatoic anhydride with ethyl acetoacetate: preparation of ethyl 4-hydroxy-2-methylquinoline-3-carboxylate and derivatives
- Nicholas G. Jentsch,
- Jared D. Hume,
- Emily B. Crull,
- Samer M. Beauti,
- Amy H. Pham,
- Julie A. Pigza,
- Jacques J. Kessl and
- Matthew G. Donahue
Beilstein J. Org. Chem. 2018, 14, 2529–2536, doi:10.3762/bjoc.14.229
Design and synthesis of C3-symmetric molecules bearing propellane moieties via cyclotrimerization and a ring-closing metathesis sequence
- Sambasivarao Kotha,
- Saidulu Todeti and
- Vikas R. Aswar
Beilstein J. Org. Chem. 2018, 14, 2537–2544, doi:10.3762/bjoc.14.230
Synthesis of 3-aminocoumarin-N-benzylpyridinium conjugates with nanomolar inhibitory activity against acetylcholinesterase
- Nisachon Khunnawutmanotham,
- Cherdchai Laongthipparos,
- Patchreenart Saparpakorn,
- Nitirat Chimnoi and
- Supanna Techasakul
Beilstein J. Org. Chem. 2018, 14, 2545–2552, doi:10.3762/bjoc.14.231
Learning from B12 enzymes: biomimetic and bioinspired catalysts for eco-friendly organic synthesis
- Keishiro Tahara,
- Ling Pan,
- Toshikazu Ono and
- Yoshio Hisaeda
Beilstein J. Org. Chem. 2018, 14, 2553–2567, doi:10.3762/bjoc.14.232
Carbonylonium ions: the onium ions of the carbonyl group
- Daniel Blanco-Ania and
- Floris P. J. T. Rutjes
Beilstein J. Org. Chem. 2018, 14, 2568–2571, doi:10.3762/bjoc.14.233
Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones
- Xiaochen Du,
- Jianjun Huang,
- Anton A. Nechaev,
- Ruwei Yao,
- Jing Gong,
- Erik V. Van der Eycken,
- Olga P. Pereshivko and
- Vsevolod A. Peshkov
Beilstein J. Org. Chem. 2018, 14, 2572–2579, doi:10.3762/bjoc.14.234
Impact of Pseudomonas aeruginosa quorum sensing signaling molecules on adhesion and inflammatory markers in endothelial cells
- Carmen Curutiu,
- Florin Iordache,
- Veronica Lazar,
- Aurelia Magdalena Pisoschi,
- Aneta Pop,
- Mariana Carmen Chifiriuc and
- Alina Maria Hoban
Beilstein J. Org. Chem. 2018, 14, 2580–2588, doi:10.3762/bjoc.14.235
Microwave-assisted synthesis of biologically relevant steroidal 17-exo-pyrazol-5'-ones from a norpregnene precursor by a side-chain elongation/heterocyclization sequence
- Gergő Mótyán,
- László Mérai,
- Márton Attila Kiss,
- Zsuzsanna Schelz,
- Izabella Sinka,
- István Zupkó and
- Éva Frank
Beilstein J. Org. Chem. 2018, 14, 2589–2596, doi:10.3762/bjoc.14.236
Synthesis of cis-hydrindan-2,4-diones bearing an all-carbon quaternary center by a Danheiser annulation
- Gisela V. Saborit,
- Carlos Cativiela,
- Ana I. Jiménez,
- Josep Bonjoch and
- Ben Bradshaw
Beilstein J. Org. Chem. 2018, 14, 2597–2601, doi:10.3762/bjoc.14.237
Synthesis of functionalised β-keto amides by aminoacylation/domino fragmentation of β-enamino amides
- Pavel Yanev and
- Plamen Angelov
Beilstein J. Org. Chem. 2018, 14, 2602–2606, doi:10.3762/bjoc.14.238
Pathoblockers or antivirulence drugs as a new option for the treatment of bacterial infections
- Matthew B. Calvert,
- Varsha R. Jumde and
- Alexander Titz
Beilstein J. Org. Chem. 2018, 14, 2607–2617, doi:10.3762/bjoc.14.239
Transition metal-free oxidative and deoxygenative C–H/C–Li cross-couplings of 2H-imidazole 1-oxides with carboranyl lithium as an efficient synthetic approach to azaheterocyclic carboranes
- Lidia A. Smyshliaeva,
- Mikhail V. Varaksin,
- Pavel A. Slepukhin,
- Oleg N. Chupakhin and
- Valery N. Charushin
Beilstein J. Org. Chem. 2018, 14, 2618–2626, doi:10.3762/bjoc.14.240
Targeting the Pseudomonas quinolone signal quorum sensing system for the discovery of novel anti-infective pathoblockers
- Christian Schütz and
- Martin Empting
Beilstein J. Org. Chem. 2018, 14, 2627–2645, doi:10.3762/bjoc.14.241
The design and synthesis of an antibacterial phenothiazine–siderophore conjugate
- Abed Tarapdar,
- James K. S. Norris,
- Oliver Sampson,
- Galina Mukamolova and
- James T. Hodgkinson
Beilstein J. Org. Chem. 2018, 14, 2646–2650, doi:10.3762/bjoc.14.242
Non-native autoinducer analogs capable of modulating the SdiA quorum sensing receptor in Salmonella enterica serovar Typhimurium
- Matthew J. Styles and
- Helen E. Blackwell
Beilstein J. Org. Chem. 2018, 14, 2651–2664, doi:10.3762/bjoc.14.243
Novel solid-phase strategy for the synthesis of ligand-targeted fluorescent-labelled chelating peptide conjugates as a theranostic tool for cancer
- Sagnik Sengupta,
- Mena Asha Krishnan,
- Premansh Dudhe,
- Ramesh B. Reddy,
- Bishnubasu Giri,
- Sudeshna Chattopadhyay and
- Venkatesh Chelvam
Beilstein J. Org. Chem. 2018, 14, 2665–2679, doi:10.3762/bjoc.14.244
Synthesis and biological evaluation of 1,2-disubstituted 4-quinolone analogues of Pseudonocardia sp. natural products
- Stephen M. Geddis,
- Teodora Coroama,
- Suzanne Forrest,
- James T. Hodgkinson,
- Martin Welch and
- David R. Spring
Beilstein J. Org. Chem. 2018, 14, 2680–2688, doi:10.3762/bjoc.14.245
Assembly of fully substituted triazolochromenes via a novel multicomponent reaction or mechanochemical synthesis
- Robby Vroemans,
- Yenthel Verhaegen,
- My Tran Thi Dieu and
- Wim Dehaen
Beilstein J. Org. Chem. 2018, 14, 2689–2697, doi:10.3762/bjoc.14.246
Ring-opening metathesis of some strained bicyclic systems; stereocontrolled access to diolefinated saturated heterocycles with multiple stereogenic centers
- Zsanett Benke,
- Melinda Nonn,
- Márton Kardos,
- Santos Fustero and
- Loránd Kiss
Beilstein J. Org. Chem. 2018, 14, 2698–2707, doi:10.3762/bjoc.14.247
